TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 119nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Inhibition of MRP1 in human COR-L23/R cells assessed reduction in tritiated daunomycin efflux incubated for 2 hrs by radioactivity-based assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 133nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 146nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 147nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 151nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 156nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 169nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 188nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 189nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 202nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2 cells co-expressing BCRP (unknown origin) assessed as effect on pheophorbide A accumulation p...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2-BCRP cells assessed as reduction in pheophorbide A accumulation measured after 120 mins by fl...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 223nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 253nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2-BCRP cells preincubated for 30 mins followed by Hoechst 33342 addition and measured at 60 sec...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 271nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 274nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 274nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 283nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 293nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 307nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 30 mins followed by Hoechst 33342 addition and measured every 6...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 312nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 322nMAssay Description:Inhibition of ABCC1 in human H69AR cells preincubated for 30 mins followed by calcein-AM addition measured at 60 secs time interval by fluorescence a...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 328nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 373nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 385nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 386nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 387nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 416nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 435nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK-II cells assessed as reduction in pheophorbide A efflux measured after 2 hrs by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 503nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 516nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in MDCK2-BCRP cells assessed as reduction in pheophorbide A accumulation measured after 120 mins by fl...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-University Bonn
Curated by ChEMBL
Affinity DataIC50: 544nMAssay Description:Inhibition of human ABCG2 expressed in MDCK2 cells co-expressing GFP preincubated for 15 mins followed by pheophorbideA addition and measured after 2...More data for this Ligand-Target Pair