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Found 31 with Last Name = 'stefan laufer' and Initial = 'na'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253323(2-(4-(4-Fluorophenyl)-5-(2-(tetrahydro-2H-pyran-4-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253374((1R,4R)-4-(4-(4-(4-Fluorophenyl)-2-(2-hydroxyethyl...)
Affinity DataIC50:  2nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253945((2S)-3-(4-(4-Fluorophenyl)-5-(2-(isopropylamino)py...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253907(3-(4-(4-Fluorophenyl)-5-(2-(tetrahydro-2H-pyran-4-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253322(2-(4-(4-Fluorophenyl)-5-(2-(isopropylamino)pyridin...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253906(3-(4-(4-Fluorophenyl)-5-(2-(isopropylamino)pyridin...)
Affinity DataIC50:  3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253503(CHEMBL522486 | Methyl 2-(4-(4-Fluorophenyl)-5-(2-(...)
Affinity DataIC50:  4nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253905(3-(4-(4-Fluorophenyl)-5-(2-(sec-butylamino)pyridin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50251985(4-(4-(4-fluorophenyl)-2-(methylthio)-1H-imidazol-5...)
Affinity DataIC50:  5nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253944((2R)-3-(4-(4-Fluorophenyl)-5-(2-(isopropylamino)py...)
Affinity DataIC50:  6nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253943((2S)-3-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-y...)
Affinity DataIC50:  10nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253320(2-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-ylamin...)
Affinity DataIC50:  11nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253946(3-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-ylamin...)
Affinity DataIC50:  12nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253867(3-(4-(4-Fluorophenyl)-5-(2-(isobutylamino)pyridin-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253904(3-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-ylamin...)
Affinity DataIC50:  15nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253942((2R)-3-(4-(4-Fluorophenyl)-5-(2-(3-methylbutan-2-y...)
Affinity DataIC50:  18nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253321(CHEMBL492295 | Methyl 2-(4-(4-Fluorophenyl)-5-(2-(...)
Affinity DataIC50:  19nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253868(3-(5-(2-(Ethylamino)pyridin-4-yl)-4-(4-fluoropheny...)
Affinity DataIC50:  27nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253500(CHEMBL492264 | Methyl 2-(4-(4-Fluorophenyl)-5-(2-(...)
Affinity DataIC50:  36nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253501(2-(4-(4-Fluorophenyl)-5-(2-(1-phenylethylamino)pyr...)
Affinity DataIC50:  37nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253865(3-(4-(4-Fluorophenyl)-5-(2-(1-phenylethylamino)pyr...)
Affinity DataIC50:  41nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253866(3-(5-(2-(1-Benzylamino)pyridin-4-yl)-4-(4-fluoroph...)
Affinity DataIC50:  87nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253903(3-(4-(4-Fluorophenyl)-5-(2-(methylamino)pyridin-4-...)
Affinity DataIC50:  102nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253831(CHEMBL505334 | Methyl 2-(4-(4-Fluorophenyl)-5-(pyr...)
Affinity DataIC50:  158nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253829(2-(4-(4-Fluorophenyl)-5-(pyridin-4-yl)-1H-imidazol...)
Affinity DataIC50:  184nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253828(3-(4-(4-Fluorophenyl)-5-(pyridin-4-yl)-1H-imidazol...)
Affinity DataIC50:  215nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253791(3-(4-(4-Fluorophenyl)-5-(pyridin-4-yl)-1H-imidazol...)
Affinity DataIC50:  392nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253502(CHEMBL492463 | Diethyl (4-(4-Fluorophenyl)-5-(2-(1...)
Affinity DataIC50:  400nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253830(CHEMBL516620 | Methyl 4-(4-(4-Fluorophenyl)-5-(pyr...)
Affinity DataIC50:  487nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253864(3-(4-(4-Fluorophenyl)-1-methyl-5-(pyridin-4yl)-1H-...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard-Karls University Of TüBingen

Curated by ChEMBL
LigandPNGBDBM50253827(CHEMBL518798 | Diethyl 2-4(4-(4-Fluorophenyl)-5-(p...)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of p38alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed