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Found 33 with Last Name = 'stempka' and Initial = 'm'
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318713((2S,15S,18S,21S,24S)-15-(3-amino-3-oxopropyl)-2-be...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314131((S,E)-Ethyl 4-((R)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  140nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314126((S)-Benzyl-2-[(Z)-3-((S)-1-benzyloxycarbonyl-2-phe...)
Affinity DataKi:  150nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  200nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assay in presence of de...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318714((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314130((S)-2-[(E)-3-((S)-1-Benzyloxycarbonyl-2-phenylethy...)
Affinity DataKi:  340nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assay in presence of d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318711((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  400nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  470nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using low concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314125((S,E)-Ethyl 4-((S)-2-(tert-Butoxycarbonylamino)-2-...)
Affinity DataKi:  640nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain using high concentration of enzyme by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318715((2S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,21-d...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318716((2S,8S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,2...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314127((S)-Benzyl-2-{(Z)-3-[(S)-1-((S)-1-benzyloxycarbony...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314128((S,E)-Methyl 2-(4-Ethoxy-4-oxobut-2-enamido)-5-oxo...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318717((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318709((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314124((S,E)-ethyl 4-(tert-butoxycarbonylamino)-7-oxo-7-(...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assay in presence of DTTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314124((S,E)-ethyl 4-(tert-butoxycarbonylamino)-7-oxo-7-(...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314132((2S,5S,8S,11S,E)-1-Benzyl 16-ethyl 11-(3-amino-3-o...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50314129((S,E)-3-((S)-1-Benzyloxycarbonyl-2-phenylethylcarb...)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense recombinant rhodesain by standard fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318714((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318718((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  2.08E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318711((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  2.22E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  2.29E+4nMAssay Description:Inhibition of human liver cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318715((2S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,21-d...)
Affinity DataKi:  3.07E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318716((2S,8S,15S,18S,21S,24S)-2-benzyl-24-carbamoyl-18,2...)
Affinity DataKi:  3.36E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318710((2S,15S,18S,21S,24S)-2,15-dibenzyl-24-carbamoyl-18...)
Affinity DataKi:  3.48E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318712((2S,15S,18S,21S,24S)-15-(2-amino-2-oxoethyl)-2-ben...)
Affinity DataKi:  3.75E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Bos taurus (bovine))
University Of Duisburg-Essen

Curated by ChEMBL
LigandPNGBDBM50318717((2S,15S,18S,21S,24S)-15-(acetamidomethyl)-2-benzyl...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of bovine spleen cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed