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TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497388(US11007200, Example 4a | US11426411, Example 4a)
Affinity DataKi:  15.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497388(US11007200, Example 4a | US11426411, Example 4a)
Affinity DataKi:  15.5nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497384(US11007200, Example 2a | US11426411, Example 2a)
Affinity DataKi:  17.3nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497384(US11007200, Example 2a | US11426411, Example 2a)
Affinity DataKi:  17.3nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497386(US11007200, Example 3a | US11426411, Example 3a)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497386(US11007200, Example 3a | US11426411, Example 3a)
Affinity DataKi:  18nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497386(US11007200, Example 3a | US11426411, Example 3a)
Affinity DataKi:  35.4nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497386(US11007200, Example 3a | US11426411, Example 3a)
Affinity DataKi:  35.4nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM568457(US11426411, Example 2b)
Affinity DataKi:  37.2nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497391(US11007200, Example 2b)
Affinity DataKi:  37.2nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497384(US11007200, Example 2a | US11426411, Example 2a)
Affinity DataKi:  59.8nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497384(US11007200, Example 2a | US11426411, Example 2a)
Affinity DataKi:  59.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497390(US11007200, Example 13a | US11426411, Example 13a)
Affinity DataKi:  70nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497390(US11007200, Example 13a | US11426411, Example 13a)
Affinity DataKi:  70nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497388(US11007200, Example 4a | US11426411, Example 4a)
Affinity DataKi:  97.2nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497388(US11007200, Example 4a | US11426411, Example 4a)
Affinity DataKi:  97.2nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497390(US11007200, Example 13a | US11426411, Example 13a)
Affinity DataKi:  98nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497390(US11007200, Example 13a | US11426411, Example 13a)
Affinity DataKi:  98nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105135(CHEMBL542936 | N2-(3-((12-((3-((4Amino,6-(methylam...)
Affinity DataKi:  135nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497392(US11007200, Example 13b | US11426411, Example 13b)
Affinity DataKi:  146nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497392(US11007200, Example 13b | US11426411, Example 13b)
Affinity DataKi:  146nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497387(US11007200, Example 3b | US11426411, Example 3b)
Affinity DataKi:  217nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497387(US11007200, Example 3b | US11426411, Example 3b)
Affinity DataKi:  217nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105123(CHEMBL544581 | N2-(3-((12-((3-((4Amino,6-(dimethyl...)
Affinity DataKi:  240nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497391(US11007200, Example 2b)
Affinity DataKi:  305nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM568457(US11426411, Example 2b)
Affinity DataKi:  305nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105120(CHEMBL542932 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  410nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497389(US11007200, Example 4b | US11426411, Example 4b)
Affinity DataKi:  426nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497389(US11007200, Example 4b | US11426411, Example 4b)
Affinity DataKi:  426nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497392(US11007200, Example 13b | US11426411, Example 13b)
Affinity DataKi:  435nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497392(US11007200, Example 13b | US11426411, Example 13b)
Affinity DataKi:  435nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105124(CHEMBL553117 | N2-(3-[12-(3-[(4,6-Diamino-1,3,5-tr...)
Affinity DataKi:  500nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105137(CHEMBL545281 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  600nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497387(US11007200, Example 3b | US11426411, Example 3b)
Affinity DataKi:  675nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma intracellular receptor 2(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497387(US11007200, Example 3b | US11426411, Example 3b)
Affinity DataKi:  675nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497389(US11007200, Example 4b | US11426411, Example 4b)
Affinity DataKi:  697nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Medisynergics

US Patent
LigandPNGBDBM497389(US11007200, Example 4b | US11426411, Example 4b)
Affinity DataKi:  697nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105121(CHEMBL542204 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  750nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105125(CHEMBL541322 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  1.00E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105139(CHEMBL544580 | N1,N9-Di(3-(((4,6-(dimethylamino-1,...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105132(CHEMBL544335 | N2-(3-((12-((3-((4,6-Di(dimethylami...)
Affinity DataKi:  2.50E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105141(CHEMBL542698 | N2-(3-((12-((3-((4,6-Di(methylamino...)
Affinity DataKi:  3.20E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105133(CHEMBL541581 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  4.60E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105134(CHEMBL555240 | N1,N9-Di(3-(di((4,6-diamino-1,3,5-t...)
Affinity DataKi:  6.70E+3nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105119(CHEMBL539797 | N2-(3-((9-((3-((4-Amino-6-(methylam...)
Affinity DataKi:  1.00E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105129(CHEMBL542208 | N2-(3-((9-((3-((4,6-Di(methylamino)...)
Affinity DataKi:  1.40E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105118(CHEMBL536324 | N1,N9-Di(3-(((4-amino-6-(dimethylam...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105142(CHEMBL554895 | N-{3-[9-(3-Amino-propylamino)-nonyl...)
Affinity DataKi:  1.70E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105138(CHEMBL543641 | N2-(3-[9-(3-[(4,6-Diamino-1,3,5-tri...)
Affinity DataKi:  1.90E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine transporter 1(Trypanosoma brucei)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50105128(CHEMBL538778 | N-{3-[12-(3-Amino-propylamino)-dode...)
Affinity DataKi:  2.50E+4nMAssay Description:Ability to inhibit adenosine uptake by the P2 transporter in Trypanosoma bruceiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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