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Found 107 with Last Name = 'steyaert' and Initial = 'j'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454561(CHEMBL4214185)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371003(CHEMBL397507)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454561(CHEMBL4214185)
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454558(CHEMBL4217119)
Affinity DataKi:  4.39E+3nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50234567(1,4-dideoxy-1,4-imino-D-ribitol | CHEMBL261634 | I...)
Affinity DataKi:  6.10E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260497(1,4-Dideoxy-1,4-imino-N-(4-amidinobenzyl)-D-ribito...)
Affinity DataKi:  6.70E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260496(1,4-Dideoxy-1,4-imino-N-(4-guanidinobenzyl)-D-ribi...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454560(CHEMBL4218602)
Affinity DataKi:  7.89E+3nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454564(CHEMBL4209269)
Affinity DataKi:  1.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260490((1S )-1,4-Dideoxy-1-(2-guanidinoethyl)-1,4-imino-D...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454554(CHEMBL4209786)
Affinity DataKi:  2.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370996(CHEMBL230908)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370998(CHEMBL397508)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454564(CHEMBL4209269)
Affinity DataKi:  2.50E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371000(CHEMBL231322)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454559(CHEMBL4202934)
Affinity DataKi:  3.35E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454557(CHEMBL4214761)
Affinity DataKi:  3.38E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454554(CHEMBL4209786)
Affinity DataKi:  3.62E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260492(1,4-Dideoxy-(3-guanidinopropyl)-1,4-imino-D-ribito...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50037773(CHEMBL3358195)
Affinity DataKi:  4.32E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454563(CHEMBL4204907)
Affinity DataKi:  5.23E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50377915(CHEMBL1169558)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371001(CHEMBL395797)
Affinity DataKi:  6.30E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454560(CHEMBL4218602)
Affinity DataKi:  7.40E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454565(CHEMBL4210507)
Affinity DataKi:  7.81E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454562(CHEMBL4208846)
Affinity DataKi:  8.04E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454562(CHEMBL4208846)
Affinity DataKi:  8.38E+4nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50371002(CHEMBL230061)
Affinity DataKi:  8.70E+4nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454553(CHEMBL4202968)
Affinity DataKi:  9.54E+4nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454558(CHEMBL4217119)
Affinity DataKi:  2.68E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260491(1,4-Dideoxy-(2-guanidinoethyl)-1,4-imino-D-ribitol...)
Affinity DataKi:  2.86E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260487(1-Guanidino-3,6-anhydro-1,2-dideoxy-Dallo-heptitol...)
Affinity DataKi:  3.09E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454559(CHEMBL4202934)
Affinity DataKi:  3.65E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50037773(CHEMBL3358195)
Affinity DataKi:  3.73E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454563(CHEMBL4204907)
Affinity DataKi:  3.93E+5nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370999(CHEMBL231025)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260486(1-Guanidino-2,5-anhydro-1-deoxy-D-allitol | CHEMBL...)
Affinity DataKi:  5.45E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260489(1-Guanidino-4,7-anhydro-1,2,3-trideoxy-Dallo-octit...)
Affinity DataKi:  6.77E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50370997(CHEMBL425996)
Affinity DataKi:  6.80E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260488(2-Guanidino-4,7-anhydro-1,2,3-trideoxy-Dallo-octit...)
Affinity DataKi:  6.85E+5nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454557(CHEMBL4214761)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454552(CHEMBL4213668)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454565(CHEMBL4210507)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454552(CHEMBL4213668)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb80-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Philipps-University Marburg

Curated by ChEMBL
LigandPNGBDBM50454553(CHEMBL4202968)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]-DHA from Nb69-fused beta2 adrenergic receptor (unknown origin) expressed in Sf9 cell membranes after 2 hrs by microbeta scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260485(2,5-Anhydro-1-deoxy-1-(trimethylammonio)-D-allitol...)
Affinity DataKi:  1.28E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50260480((2R,3S,4R,5R)-3,4-Dihydroxy-5-(hydroxymethyl)-tetr...)
Affinity DataKi:  4.50E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50206267((2S,3R,4S,5R)-2-(2-azidoethyl)-5-(hydroxymethyl)-t...)
Affinity DataKi:  5.60E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIAG-nucleoside hydrolase(Trypanosoma vivax)
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50206267((2S,3R,4S,5R)-2-(2-azidoethyl)-5-(hydroxymethyl)-t...)
Affinity DataKi:  5.64E+6nMAssay Description:Inhibition of Trypanosoma vivax IAG-nucleoside hydrolase expressed in Escherichia coli WK6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Homo sapiens (Human))
Galapagos

Curated by ChEMBL
LigandPNGBDBM50257775(CHEMBL4100462)
Affinity DataIC50:  2nMAssay Description:Inhibition of glycosylated human ATX using FS-3 as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by fluore...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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