Affinity DataKi: 0.0631nMAssay Description:Effect on pancreatic polypeptide-mediated displacement of 125I-pancreatic polypeptide from human C-terminal eYFP-tagged NY4 receptor expressed in HEK...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Effect on peptide YY-mediated displacement of 125I-pancreatic polypeptide from human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cell mem...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Effect on neuropeptide Y-mediated displacement of 125I-pancreatic polypeptide from human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cell...More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Allosteric antagonist activity at NPY5R in mouse descending colon mucosa assessed as reduction in rPP-induced ion transport by electrophysiologyMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Allosteric antagonist activity at NPY5R in mouse descending colon mucosa assessed as reduction in rPP-induced ion transport by electrophysiologyMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Allosteric antagonist activity at eFYP-tagged human NPY4R expressed in COS7 cells co-expressing Gqi5-alpha assessed as inhibition of PP-induced Ca2+ ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0398nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY1 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0631nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY2 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY5 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
Affinity DataEC50: 845nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of peptide YY-induced ...More data for this Ligand-Target Pair
Affinity DataEC50: 0.501nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of neuropeptide Y-indu...More data for this Ligand-Target Pair
Affinity DataEC50: 5.01E+3nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 9nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 280nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 564nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 966nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 195nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 282nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 955nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Agonist activity at wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as increase in calcium flux measured for 40 sec by Fluo-2 AM d...More data for this Ligand-Target Pair
Affinity DataEC50: 134nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 513nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 150nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 135nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 513nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 151nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-fused human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Gal...More data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of peptide YY-induced ...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of pancreatic polypept...More data for this Ligand-Target Pair
Affinity DataEC50: 0.398nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0398nMAssay Description:Positive allosteric modulation of human NY4 receptor expressed in African green monkey COS7 cells co-expressing delta6Galphaqi4-myr assessed as poten...More data for this Ligand-Target Pair
Affinity DataEC50: 443nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of neuropeptide Y-indu...More data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Positive allosteric modulation of human C-terminal eYFP-tagged NY4 receptor expressed in HEK293 cells assessed as potentiation of pancreatic polypept...More data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at Wild type CMKL1 (unknown origin) expressed in COS-7 cells assessed as accumulation of inositol phosphate incubated for 3 hrs by l...More data for this Ligand-Target Pair