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Found 15 with Last Name = 'stockwell' and Initial = 'br'
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126160(CHEMBL3629669)
Affinity DataIC50:  4nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126159(CHEMBL3629668)
Affinity DataIC50:  10nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126156(CHEMBL3629579)
Affinity DataIC50:  10nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126155(CHEMBL3629578)
Affinity DataIC50:  20nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126162(CHEMBL3629671)
Affinity DataIC50:  30nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126153(CHEMBL3629576)
Affinity DataIC50:  30nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126154(CHEMBL3629577)
Affinity DataIC50:  40nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126152(CHEMBL3629575)
Affinity DataIC50:  60nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50593519(CHEMBL5204252)
Affinity DataIC50:  96nMAssay Description:Inhibition of chymotrypsin-like activity of human erythrocytes 20S proteasome using Suc-LLVY-AMC as substrate and measured by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126161(CHEMBL3629670)
Affinity DataIC50:  100nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50376126(ERASTIN)
Affinity DataIC50:  200nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126157(CHEMBL3629580)
Affinity DataIC50:  300nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystine/glutamate transporter(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50126151(CHEMBL3629574)
Affinity DataIC50:  800nMAssay Description:Inhibition of Xct in human CCF-STTG1 cells assessed as glutamate release after 2 hrs by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50499156(CHEMBL1358404)
Affinity DataKd:  7.58E+5nMAssay Description:Binding affinity to PDI catalytic domain a (unknown origin) after 1 hrs by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent anion-selective channel protein 2(Homo sapiens (Human))
Columbia University

Curated by ChEMBL
LigandPNGBDBM50376126(ERASTIN)
Affinity DataKd:  100nMAssay Description:Binding affinity to human VDAC2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed