Affinity DataKi: 6nM ΔG°: -48.8kJ/mole IC50: 32nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 8.5nMAssay Description:Activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 9nM ΔG°: -47.8kJ/mole IC50: 51nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 11nM ΔG°: -47.3kJ/mole IC50: 60nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Activity at CB2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nM ΔG°: -46.8kJ/mole IC50: 73nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 19nM ΔG°: -45.8kJ/mole IC50: 107nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 20nM ΔG°: -45.7kJ/mole IC50: 112nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 26nM ΔG°: -45.0kJ/mole IC50: 146nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 28nM ΔG°: -44.8kJ/mole IC50: 154nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 40nM ΔG°: -43.9kJ/mole IC50: 222nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 41nM ΔG°: -43.9kJ/mole IC50: 231nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 44nM ΔG°: -43.7kJ/mole IC50: 245nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 46nM ΔG°: -43.6kJ/mole IC50: 255nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 49nM ΔG°: -43.4kJ/mole IC50: 271nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 53nM ΔG°: -43.2kJ/mole IC50: 297nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 58nM ΔG°: -43.0kJ/mole IC50: 325nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 81nM ΔG°: -42.1kJ/mole IC50: 454nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 104nM ΔG°: -41.5kJ/mole IC50: 580nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 111nM ΔG°: -41.3kJ/mole IC50: 619nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 160nM ΔG°: -40.3kJ/mole IC50: 891nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 2.07E+3nM ΔG°: -33.7kJ/mole IC50: 1.16E+4nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nM ΔG°: -31.7kJ/mole IC50: 2.57E+4nMpH: 9.5 T: 2°CAssay Description:Inhibition of WNV protease activity was measured using recombinant WNV protease, which first incubated with inhibitor in 96-well plates. Catalysis wa...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataIC50: 0.320nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Agonist activity at CB1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 6.31nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
The University Of Queensland
Curated by ChEMBL
The University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-C3a from C3AR in HMDMs by scintillation counting methodMore data for this Ligand-Target Pair