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Found 195 with Last Name = 'stroke' and Initial = 'il'
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454459(CHEMBL4215036)
Affinity DataIC50:  1nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454459(CHEMBL4215036)
Affinity DataIC50:  1nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507130(CHEMBL4452983)
Affinity DataIC50:  2nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507108(CHEMBL4529863)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454497(CHEMBL4214079)
Affinity DataIC50:  3nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454500(CHEMBL4212258)
Affinity DataIC50:  3nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507128(CHEMBL4451752)
Affinity DataIC50:  4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507134(CHEMBL4444965)
Affinity DataIC50:  4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507115(CHEMBL4520413)
Affinity DataIC50:  4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507107(CHEMBL4473557)
Affinity DataIC50:  4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507135(CHEMBL4470638)
Affinity DataIC50:  4nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507120(CHEMBL4473443)
Affinity DataIC50:  5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507105(CHEMBL4557223)
Affinity DataIC50:  5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507127(CHEMBL4476228)
Affinity DataIC50:  5nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507133(CHEMBL4461315)
Affinity DataIC50:  6nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507136(CHEMBL4454294)
Affinity DataIC50:  7nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454497(CHEMBL4214079)
Affinity DataIC50:  7nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507126(CHEMBL4483028)
Affinity DataIC50:  8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507114(CHEMBL4553525)
Affinity DataIC50:  8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507113(CHEMBL4436890)
Affinity DataIC50:  8nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454486(CHEMBL4203819)
Affinity DataIC50:  9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507116(CHEMBL4452876)
Affinity DataIC50:  9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507119(CHEMBL4441033)
Affinity DataIC50:  9nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507106(CHEMBL4472977)
Affinity DataIC50:  10nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507129(CHEMBL4456814)
Affinity DataIC50:  14nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507112(CHEMBL4547929)
Affinity DataIC50:  18nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454504(CHEMBL4210388)
Affinity DataIC50:  18nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50413094(CHEMBL486116)
Affinity DataIC50:  18.6nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50413093(CHEMBL528990)
Affinity DataIC50:  19.5nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175173(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CXCL10(IP-10)-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507118(CHEMBL4456808)
Affinity DataIC50:  20nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507117(CHEMBL4591470)
Affinity DataIC50:  21nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507105(CHEMBL4557223)
Affinity DataIC50:  24nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50413092(CHEMBL519258)
Affinity DataIC50:  25.1nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507135(CHEMBL4470638)
Affinity DataIC50:  29nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507109(CHEMBL4530206)
Affinity DataIC50:  38nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507121(CHEMBL4589634)
Affinity DataIC50:  41nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454503(CHEMBL4211420)
Affinity DataIC50:  42nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454498(CHEMBL4215657)
Affinity DataIC50:  43nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507110(CHEMBL4545776)
Affinity DataIC50:  45nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B glucosyltransferase domain assessed as reduction in UDP-glucose hydro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50454502(CHEMBL4209041)
Affinity DataIC50:  50nMAssay Description:Inhibition of C-terminal 6-His tagged recombinant Clostridium difficile toxin B catalytic fragment (Met1 to Leu543 residues) assessed as reduction in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175193(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)
Affinity DataIC50:  50nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Pharmacopeia

Curated by ChEMBL
LigandPNGBDBM50413100(CHEMBL485915)
Affinity DataIC50:  51.3nMAssay Description:Antagonist activity at human OX2 receptor expressed in HEK293 cells assessed as inhibition of human orexin-A-stimulated calcium release by FLIPR assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507114(CHEMBL4553525)
Affinity DataIC50:  52nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToxin B(Peptoclostridium difficile)
Genesis Biotechnology Group

Curated by ChEMBL
LigandPNGBDBM50507115(CHEMBL4520413)
Affinity DataIC50:  53nMAssay Description:Inhibition of Clostridium difficile toxin B transfected in CHO cells assessed as reduction in caspase 3/7 activation pre-incubated for 1 hr before Tc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175183(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)
Affinity DataIC50:  60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175168(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)
Affinity DataIC50:  60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175176(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-fluor...)
Affinity DataIC50:  60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50175173(4-(4-((2,4-dichlorophenethyl)carbamoyl)-2-(3-chlor...)
Affinity DataIC50:  60nMAssay Description:Inhibition of CXCL11-stimulated calcium release in HEK293 cells expressing recombinant human CXCR3 and chimeric G protein Gqi5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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