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Found 50 with Last Name = 'strosberg' and Initial = 'am'
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.603nMAssay Description:Affinity for alpha-1 adrenoceptor of rat cerebral cortex was determined by ligand binding using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50033113(CHEMBL279516 | INDORAMIN | INDORAMINE | INDORAMINN...)
Affinity DataKi:  25nMAssay Description:Affinity for alpha-1 adrenoceptor of rat cerebral cortex was determined by ligand binding using [3H]prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50224806(CHEMBL355655)
Affinity DataKi:  39nMAssay Description:Affinity for alpha-1 adrenoceptor of rat cerebral cortex was determined by ligand binding using [3H]prazosin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50224806(CHEMBL355655)
Affinity DataKi:  631nMAssay Description:Affinity for alpha-2 adrenergic receptor of rat cerebral cortex was determined by ligand binding using [3H]yohimbine.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  646nMAssay Description:Affinity for alpha-2 adrenergic receptor of rat cerebral cortex was determined by ligand binding using [3H]yohimbineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50033113(CHEMBL279516 | INDORAMIN | INDORAMINE | INDORAMINN...)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity for alpha-2 adrenergic receptor of rat cerebral cortex was determined by ligand binding using [3H]yohimbine.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227226(CHEMBL68378)
Affinity DataIC50:  5nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000871(CHEMBL69139 | N-Cyclohexyl-N-methyl-4-(2-oxo-1,2,3...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227219(CHEMBL68848)
Affinity DataIC50:  6.10nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227212(CHEMBL308196)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227216(CHEMBL69307)
Affinity DataIC50:  9.30nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000871(CHEMBL69139 | N-Cyclohexyl-N-methyl-4-(2-oxo-1,2,3...)
Affinity DataIC50:  10nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227222(CHEMBL66973)
Affinity DataIC50:  10nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227214(CHEMBL68708)
Affinity DataIC50:  16nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227218(CHEMBL305411)
Affinity DataIC50:  35nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227227(CHEMBL305979)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227221(CHEMBL302724)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227224(CHEMBL67246)
Affinity DataIC50:  60nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227211(CHEMBL302079)
Affinity DataIC50:  63nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227206(CHEMBL66522)
Affinity DataIC50:  70nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000334(6,7-Dichloro-1,5-dihydro-imidazo[2,1-b]quinazolin-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227228(CHEMBL422230)
Affinity DataIC50:  100nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227220(CHEMBL69524)
Affinity DataIC50:  120nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227195(CHEMBL31580)
Affinity DataIC50:  150nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50225945(CI-930)
Affinity DataIC50:  150nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227217(CHEMBL302049)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227207(Quazinone | Ro-136438 | Ro-136438006)
Affinity DataIC50:  240nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50226555(CHEMBL67513)
Affinity DataIC50:  290nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227215(CHEMBL66995)
Affinity DataIC50:  430nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227225(CHEMBL66845)
Affinity DataIC50:  470nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227200(CHEMBL66978)
Affinity DataIC50:  520nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227199(CHEMBL66447)
Affinity DataIC50:  560nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227194(CHEMBL66153)
Affinity DataIC50:  600nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227196(CHEMBL66061)
Affinity DataIC50:  700nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM15296(6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin...)
Affinity DataIC50:  860nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50226542(CHEMBL65882)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227204(CHEMBL66212)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227203(CHEMBL70033)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227223(CHEMBL67567)
Affinity DataIC50:  3.10E+3nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227201(CHEMBL69286)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227213(CHEMBL67392)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227208(CHEMBL65700)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227209(CHEMBL302575)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227210(CHEMBL68998)
Affinity DataIC50:  1.85E+4nMAssay Description:In vitro inhibitory activity against platelet phosphodiesterase (PDE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227205(CHEMBL66935)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227197(CHEMBL69940)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50226873(CHEMBL428866)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50225502(MDL-19205 | Piroximone)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227202(CHEMBL68833)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50227198(CHEMBL307996)
Affinity DataIC50:  3.30E+5nMAssay Description:Inhibition of platelet cAMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed