Compile Data Set for Download or QSAR
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Found 46 with Last Name = 'stuttle' and Initial = 'k'
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054959((4aS,4bR,5S,6aS,6bR,9aR)-4b-Fluoro-5-hydroxy-4a,6a...)
Affinity DataIC50:  1.60nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054966((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  1.70nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407988(CHEMBL2112857)
Affinity DataIC50:  1.80nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054953((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  2.10nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054964((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-6b-...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054961((4aS,4bR,5S,6aS,6bR,9aR,12S)-4b,12-Difluoro-5-hydr...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054955((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-5-h...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50369181(TIPREDANE)
Affinity DataIC50:  2.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054960((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-5-h...)
Affinity DataIC50:  2.40nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50354850(BUDESONIDE | US10869929, Compound Budesonide | US1...)
Affinity DataIC50:  2.90nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054952((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-6b...)
Affinity DataIC50:  3.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054963((4aS,4bR,5S,6aS,6bR,8R,9aR)-6b-Ethylsulfanyl-4b-fl...)
Affinity DataIC50:  3.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054962((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-6b-fluoromet...)
Affinity DataIC50:  3.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407989(CHEMBL2112850)
Affinity DataIC50:  4.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50354849(CCI-18781 | Cutivate | FLUTICASONE PROPIONATE | Fl...)
Affinity DataIC50:  5nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407990(CHEMBL2112858)
Affinity DataIC50:  5.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054967((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-6b...)
Affinity DataIC50:  5.5nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150059(CHEMBL183215 | N-(4-Methyl-2-pyrrolidin-1-yl-quino...)
Affinity DataIC50:  10nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054957((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  12nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054951((4aS,4bR,5S,6aS,6bR,9aR)-4b-Fluoro-5-hydroxy-4a,6a...)
Affinity DataIC50:  22nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150063(CHEMBL364863 | N-[4-Methyl-2-(4-methyl-piperazin-1...)
Affinity DataIC50:  63nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50:  71nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150064(CHEMBL182886 | N-(4-Methyl-2-morpholin-4-yl-quinol...)
Affinity DataIC50:  124nMAssay Description:Tested for MCH-1 induced [Ca2+] release from CHO cells transfected with human MCH-1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150072(2-(2,3-Dichloro-phenoxy)-N-[4-methyl-2-(4-methyl-p...)
Affinity DataIC50:  201nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50:  349nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150061(CHEMBL185376 | N-(2-Isopropylamino-4-methyl-quinol...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150063(CHEMBL364863 | N-[4-Methyl-2-(4-methyl-piperazin-1...)
Affinity DataIC50:  442nMAssay Description:Inhibitory activity against human 5-HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50:  970nMAssay Description:Inhibitory activity against human 5-HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50150057(2-(4-Chloro-phenoxy)-N-[4-methyl-2-(4-methyl-piper...)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibitory activity against human 5-HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052687(CHEMBL114705 | N-[5-(3-Cyclohexyl-propionylamino)-...)
Affinity DataEC50:  1.20E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052686(CHEMBL115992 | N-{3-[(Benzo[1,3]dioxol-5-ylmethyl)...)
Affinity DataEC50:  600nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052688(CHEMBL419042 | N-[5-(3-Cyclohexyl-propionylamino)-...)
Affinity DataEC50:  2.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052685(4-Amino-N-[5-(3-cyclohexyl-propionylamino)-2-methy...)
Affinity DataEC50:  3.80E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052680(CHEMBL419763 | N-[5-(3-Cyclohexyl-propionylamino)-...)
Affinity DataEC50:  1.70E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052683(CHEMBL112449 | N-[3-((Z)-2-Cyano-2-pyridin-3-yl-vi...)
Affinity DataEC50:  1.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052682(3-Cyclohexyl-N-[3-(5-hydroxy-1H-benzoimidazol-2-yl...)
Affinity DataEC50:  700nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052681(CHEMBL114890 | N-[3-((Z)-2-Benzo[1,3]dioxol-5-yl-2...)
Affinity DataEC50:  700nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052679(CHEMBL112537 | N-[5-(3-Cyclohexyl-propionylamino)-...)
Affinity DataEC50:  2.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052678(3-Cyclohexyl-N-[4-methyl-3-(5-methyl-1H-benzoimida...)
Affinity DataEC50:  1.30E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052677(CHEMBL115779 | N-(2-Cyclohexyl-ethyl)-3-(4-hydroxy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052676(CHEMBL115304 | N-[3-(1H-Benzoimidazol-2-yl)-4-meth...)
Affinity DataEC50:  1.30E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052690(Acetic acid 4-[5-(3-cyclohexyl-propionylamino)-2-m...)
Affinity DataEC50:  2.50E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052689(CHEMBL115205 | N-[5-(4-Cyclohexyl-butyrylamino)-2-...)
Affinity DataEC50:  4.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052691(CHEMBL114199 | N-[5-(4-Cyclohexyl-butyryl)-2-methy...)
Affinity DataEC50:  2.00E+3nMAssay Description:Concentration at which one-half the maximum Low density lipoprotein receptor upregulation is observed in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052692(5-(3-Cyclohexyl-propionylamino)-N-(4-hydroxy-pheny...)
Affinity DataEC50:  7.00E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLow-density lipoprotein receptor(Homo sapiens (Human))
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50052684(CHEMBL112106 | N-[5-(3-Cyclohexyl-propionylamino)-...)
Affinity DataEC50:  7.60E+3nMAssay Description:Concentration at which one-half of the maximum Low density lipoprotein receptor is upregulated in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed