Compile Data Set for Download or QSAR
maximum 50k data
Found 16 with Last Name = 'sucholeiki' and Initial = 'i'
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of recombinant human MMP13 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM16596(4-N,6-N-bis[(4-fluoro-3-methylphenyl)methyl]pyrimi...)
Affinity DataIC50:  8nMAssay Description:Inhibition of MMP13 (unknown origin) using APMA as substrate preincubated for 15 mins followed by substrate additionMore data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM50573596(CHEMBL4846182)
Affinity DataIC50: <10nMAssay Description:Inhibition of MMP13 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256502(US9505743, 70)
Affinity DataIC50: <100nMpH: 7.6 T: 2°CAssay Description:MMP-13 inhibitor activity of the MMP inhibitors of the present invention was measured using the method of Knight (Knight, C. G. et. al, FEBS LETT. 29...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM50573597(CHEMBL4860977)
Affinity DataIC50: >100nMAssay Description:Inhibition of MMP13 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: <100nMpH: 7.6 T: 2°CAssay Description:MMP-13 inhibitor activity of the MMP inhibitors of the present invention was measured using the method of Knight (Knight, C. G. et. al, FEBS LETT. 29...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCollagenase 3(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: <100nMpH: 7.6 T: 2°CAssay Description:MMP-13 inhibitor activity of the MMP inhibitors of the present invention was measured using the method of Knight (Knight, C. G. et. al, FEBS LETT. 29...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetStromelysin-2(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human MMP10 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50:  7.40E+4nMAssay Description:Inhibition of recombinant human MMP9 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of recombinant human MMP8 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP2 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP1 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP14 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP7 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP12 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Bolderbiopath

Curated by ChEMBL
LigandPNGBDBM256500(BDBM256501 | US9505743, 44)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human MMP3 using QXL520-gamma-Abu-Pro-Cha-Abu-Smc-His-Ala-Dab(5-FAM)-Ala-Lys-NH2 as substrate measured every 5 mins for 2 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed