Compile Data Set for Download or QSAR
maximum 50k data
Found 32 with Last Name = 'sufka' and Initial = 'kj'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388008(CHEMBL2058426)
Affinity DataKi:  591nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388016(CHEMBL2058419)
Affinity DataKi:  656nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388015(CHEMBL1170237)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388014(CHEMBL2058420)
Affinity DataKi:  1.22E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388009(METHYLAPLYSINOPSIN)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388007(CHEMBL2058427)
Affinity DataKi:  2.62E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataKi:  3.03E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50387977(CHEMBL2058415)
Affinity DataKi:  5.92E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388018(CHEMBL2058416)
Affinity DataKi:  6.18E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105335(CHEMBL3597247)
Affinity DataIC50:  280nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105353(CHEMBL3597266)
Affinity DataIC50:  290nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105355(CHEMBL3597268)
Affinity DataIC50:  410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105333(CHEMBL3597245)
Affinity DataIC50:  410nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105350(CHEMBL3597264)
Affinity DataIC50:  510nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105354(CHEMBL3597267)
Affinity DataIC50:  1.12E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105348(CHEMBL3597262)
Affinity DataIC50:  1.44E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105349(CHEMBL3597263)
Affinity DataIC50:  1.77E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50230993((2S)-2-amino-5-[(N-methylcarbamimidoyl)amino]penta...)
Affinity DataIC50:  2.30E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105344(CHEMBL3597258)
Affinity DataIC50:  2.55E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105346(CHEMBL3597260)
Affinity DataIC50:  2.57E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105351(CHEMBL3597265)
Affinity DataIC50:  2.90E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105341(CHEMBL3597254)
Affinity DataIC50:  3.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105334(CHEMBL3597246)
Affinity DataIC50:  4.22E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105332(CHEMBL3597244)
Affinity DataIC50:  4.43E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105345(CHEMBL3597259)
Affinity DataIC50:  4.50E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105339(CHEMBL3597252)
Affinity DataIC50:  4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105342(CHEMBL3597256)
Affinity DataIC50:  4.51E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105347(CHEMBL3597261)
Affinity DataIC50:  4.54E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105331(CHEMBL3597241)
Affinity DataIC50:  4.62E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105340(CHEMBL3597253)
Affinity DataIC50:  4.66E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105343(CHEMBL3597257)
Affinity DataIC50:  4.86E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50105337(CHEMBL3597251)
Affinity DataIC50:  4.98E+3nMAssay Description:Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of LPS-induced iNOS activity incubated for 30 mins prior to LPS challenge me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed