Compile Data Set for Download or QSAR
maximum 50k data
Found 72 with Last Name = 'sugioka' and Initial = 'y'
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217526(CHEMBL366972)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50057477(4-(3-{3-[(4-Isobutyl-benzyl)-(4-isobutyl-phenyl)-a...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 1 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217519(CHEMBL354709)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217520(CHEMBL354645)
Affinity DataIC50:  3.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217517(CHEMBL353158)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217511(CHEMBL172342)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217506(CHEMBL170936)
Affinity DataIC50:  5.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217509(CHEMBL354731)
Affinity DataIC50:  5.90nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217508(CHEMBL367509)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217504(CHEMBL353284)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217505(CHEMBL414377)
Affinity DataIC50:  6.70nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217513(CHEMBL171658)
Affinity DataIC50:  6.80nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217528(CHEMBL353596)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217509(CHEMBL354731)
Affinity DataIC50:  7.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217505(CHEMBL414377)
Affinity DataIC50:  7.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217522(CHEMBL353394)
Affinity DataIC50:  7.80nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217507(CHEMBL171704)
Affinity DataIC50:  9.20nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217527(CHEMBL172227)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217530(CHEMBL170084)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 2(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50057477(4-(3-{3-[(4-Isobutyl-benzyl)-(4-isobutyl-phenyl)-a...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 2 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217519(CHEMBL354709)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217528(CHEMBL353596)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217514(CHEMBL369246)
Affinity DataIC50:  13nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217510(CHEMBL355387)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217512(CHEMBL169132)
Affinity DataIC50:  16nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217527(CHEMBL172227)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217506(CHEMBL170936)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217518(CHEMBL353480)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217512(CHEMBL169132)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217529(CHEMBL171719)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217510(CHEMBL355387)
Affinity DataIC50:  21nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217529(CHEMBL171719)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217516(CHEMBL354288)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50216728(CHEMBL359360)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory activity against rat testosterone 5 alpha reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217514(CHEMBL369246)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217531(CHEMBL170083)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217515(CHEMBL352350)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217513(CHEMBL171658)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50069237(4-{2-[6-(Benzhydryl-carbamoyl)-benzofuran-2-yl]-ph...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity against rat testosterone 5 alpha reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217504(CHEMBL353284)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217523(CHEMBL353168)
Affinity DataIC50:  32nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217507(CHEMBL171704)
Affinity DataIC50:  34nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50069239(4-[2-(6-{[Bis-(4-methoxy-phenyl)-methyl]-carbamoyl...)
Affinity DataIC50:  36nMAssay Description:In vitro inhibitory activity against rat testosterone 5 alpha reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rattus norvegicus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50069235(4-[2-(6-{[Bis-(4-fluoro-phenyl)-methyl]-carbamoyl}...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibitory activity against rat testosterone 5 alpha reductase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217517(CHEMBL353158)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50069235(4-[2-(6-{[Bis-(4-fluoro-phenyl)-methyl]-carbamoyl}...)
Affinity DataIC50:  50nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 1 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217520(CHEMBL354645)
Affinity DataIC50:  51nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217523(CHEMBL353168)
Affinity DataIC50:  52nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217524(CHEMBL433909)
Affinity DataIC50:  61nMAssay Description:Inhibitory activity against Neurokinin 1 (NK1) receptor from guinea pig lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1(Homo sapiens (Human))
Sankyo

Curated by ChEMBL
LigandPNGBDBM50069237(4-{2-[6-(Benzhydryl-carbamoyl)-benzofuran-2-yl]-ph...)
Affinity DataIC50:  62nMAssay Description:In vitro inhibitory activity against human Steroid 5-alpha-reductase type 1 in COS-1 cells was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 72 total ) | Next | Last >>
Jump to: