Affinity DataIC50: 0.400nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against histone deacetylase (HDAC4) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cells; Not testedMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against histone deacetylase 6 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human histone deacetylase 4 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human histone deacetylase 1 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human histone deacetylase 6 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against histone deacetylase (HDAC4) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against histone deacetylase 6 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibitory activity against histone deacetylase 6 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against histone deacetylase 8 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human histone deacetylase 8 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against histone deacetylase 8 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human histone deacetylase 1 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibitory activity against histone deacetylase 8 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against histone deacetylase 8 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibitory activity against histone deacetylases (HDAC1) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibitory activity against histone deacetylase (HDAC4) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibitory activity against histone deacetylase (HDAC4) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Inhibitory activity against histone deacetylase 6 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of human histone deacetylase 6 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against histone deacetylase (HDAC4) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human histone deacetylase 4 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of human histone deacetylase 8 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of human histone deacetylase 8 prepared from 293T cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of human histone deacetylase 4 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of human histone deacetylase 1 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition of human histone deacetylase 8 prepared from 293T cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 782nMAssay Description:Inhibitory activity against histone deacetylase 6 prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibition of human histone deacetylase 1 prepared from 293T cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 957nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
TargetHistone deacetylase 1/2/3/4/5/6/7/8/9/11/Polyamine deacetylase HDAC10(Mus musculus)
Institute Of Technology
Curated by ChEMBL
Institute Of Technology
Curated by ChEMBL
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibitory activity against histone deacetylases (HDAC) prepared from mouse melanoma B16/BL6 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of human histone deacetylase 6 prepared from 293T cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human histone deacetylase 6 prepared from 293T cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Shinshu University
Curated by ChEMBL
Shinshu University
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of FLAG-tagged full-length human recombinant DYRK1A (127 to 485 residues) expressed in Escherichia coli assessed as reduction in autophosp...More data for this Ligand-Target Pair