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Found 27 with Last Name = 'suvire' and Initial = 'f'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50298707(1-Benzyl-6-chloro-7-hydroxy-1,2,3,4-tetrahydroisoq...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50298706(1-Butyl-6-chloro-7-hydroxy-1,2,3,4-tetrahydroisoqu...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad De Valencia

Curated by ChEMBL
LigandPNGBDBM50022051(1-Phenyl-6-chloro-7-hydroxy-N-methyl-1,2,3,4-tetra...)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Wistar rat striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  480nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  2.24E+4nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190650(CHEMBL3906484)
Affinity DataIC50:  6.73E+4nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190650(CHEMBL3906484)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190649(Montanine)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190651(CHEMBL3956367)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190651(CHEMBL3956367)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190649(Montanine)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50221066((-)-lycorine | 9,10-(methylenedioxy)-3,12-didehydr...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190648(CHEMBL3889595)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190647(CHEMBL3978970)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190648(CHEMBL3889595)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50190647(CHEMBL3978970)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of electric eel AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Universidad Nacional De San Juan

Curated by ChEMBL
LigandPNGBDBM50221066((-)-lycorine | 9,10-(methylenedioxy)-3,12-didehydr...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of equine serum BuChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 5 mins by DTNB-based ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510090(CHEMBL4535730)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510090(CHEMBL4535730)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510091(CHEMBL4519542)
Affinity DataEC50:  1.69E+3nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510092(CHEMBL4593987)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510092(CHEMBL4593987)
Affinity DataEC50:  184nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510091(CHEMBL4519542)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510093(CHEMBL4466552)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARalpha expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50510094(CHEMBL4460072)
Affinity DataEC50:  991nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Valencia

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human PPARgamma expressed in African green monkey COS7 cells assessed as increase in receptor transcriptional activity by lucifer...More data for this Ligand-Target Pair