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Found 45 with Last Name = 'sweeney' and Initial = 'mt'
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099848(CHEMBL30051 | N-Hydroxy-2-naphthalen-1-yl-2-(3-tri...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099846(CHEMBL29911 | N-Hydroxy-2-(3-methoxy-phenyl)-2-(3-...)
Affinity DataIC50:  59nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099855(2-(2-Chloro-4,5-dimethoxy-phenyl)-N-hydroxy-acetam...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099849(2-(2-Fluoro-phenyl)-N-hydroxy-2-(3-trifluoromethyl...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099847(2-(3,4-Difluoro-phenyl)-N-hydroxy-2-(3-trifluorome...)
Affinity DataIC50:  690nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099856(CHEMBL29912 | N'-hydroxy-N-1-naphthyl-N-{2-[3-(tri...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099853(CHEMBL26420 | Naphthalen-1-yl-(3-trifluoromethyl-b...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099845(2-Biphenyl-4-yl-N-hydroxy-acetamide | CHEMBL30068)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102059((3R,4R)-3-[2-(5-Bromo-2-chloro-phenyl)-ethyl]-4-fl...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099857(ACETOHYDROXAMIC ACID (AHA) | AHA | Acethydroxamsae...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099852(CHEMBL29796 | Naphthalen-1-yl-(3-trifluoromethyl-b...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099851(CHEMBL27348 | N-1-naphthyl-N-{2-[3-(trifluoromethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099850(2-Naphthalen-1-yl-2-(3-trifluoromethyl-benzylamino...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099844(2-Mercapto-N-naphthalen-1-yl-N-[2-(3-trifluorometh...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus (strain Mu50 / ATCC 700699))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50099854(2-Hydroxy-N-naphthalen-1-yl-N-[2-(3-trifluoromethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Peptidyl deformylase (PDF)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102064(3-[2-(5-Bromo-2-chloro-phenyl)-vinyl]-piperidine; ...)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102057(3-[2-(5-Bromo-2-chloro-phenyl)-ethyl]-piperidine; ...)
Affinity DataIC50:  1.85E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102061(3-[2-(2,5-Dichloro-phenyl)-ethyl]-piperidine | CHE...)
Affinity DataIC50:  1.95E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102051(3-[2-(3,4-Dichloro-phenyl)-ethyl]-piperidine | CHE...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102060(3-[2-(2,6-Dichloro-phenyl)-ethyl]-piperidine | CHE...)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102056(3-[2-(3,5-Bis-trifluoromethyl-phenyl)-ethyl]-piper...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102067((3S,4S)-3-[3-(5-Bromo-2-chloro-phenyl)-propyl]-4-f...)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102052(5-(5-bromo-2-chlorobenzyl)-4-fluoro-1,2,3,6-tetrah...)
Affinity DataIC50:  4.80E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102049(5-(5-Bromo-2-chloro-benzyl)-1,2,3,6-tetrahydro-pyr...)
Affinity DataIC50:  6.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102053((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-5-guan...)
Affinity DataIC50:  7.30E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102055(4-(2-Piperidin-3-yl-ethyl)-benzonitrile | CHEMBL55...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102063(3-[2-(4-Ethoxy-phenyl)-ethyl]-piperidine | CHEMBL5...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102062(3-(5-Bromo-2-chloro-benzyl)-piperidin-4-one; hydro...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102058((3S,4S)-3-(5-Bromo-2-chloro-benzyl)-piperidin-4-ol...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102050((S)-3-(5-Bromo-2-chloro-benzyl)-piperidin-4-ol; hy...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102065(3-[2-(3-Chloro-2'-methoxy-biphenyl-4-yl)-ethyl]-pi...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102066((3S,4S)-3-(5-Bromo-2-chloro-benzyl)-4-fluoro-piper...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102068(3-Phenethyl-piperidine | CHEMBL55554)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospho-N-acetylmuramoyl-pentapeptide-transferase(Escherichia coli (strain K12))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50102054(3-[2-(2,5-Dimethyl-phenyl)-ethyl]-piperidine | CHE...)
Affinity DataIC50: >9.00E+5nMAssay Description:Inhibitory activity against accumulation of [14C]-labeled Linezolid within wild-type Escherichia coli K12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219738(5-chloro-2-(3-(morpholinosulfonyl)benzamido)benzoi...)
Affinity DataKd:  6.50E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219737(5-bromo-2-(3-(morpholinosulfonyl)benzamido)benzoic...)
Affinity DataKd:  4.80E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219739(5-methyl-2-(3-(morpholinosulfonyl)benzamido)benzoi...)
Affinity DataKd:  7.50E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219740(5-methoxy-2-(3-(morpholinosulfonyl)benzamido)benzo...)
Affinity DataKd:  8.10E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219741(5-cyano-2-(4-(morpholinosulfonyl)benzamido)benzoic...)
Affinity DataKd:  1.40E+4nMAssay Description:Binding to high affinity site of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219741(5-cyano-2-(4-(morpholinosulfonyl)benzamido)benzoic...)
Affinity DataKd:  5.30E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219741(5-cyano-2-(4-(morpholinosulfonyl)benzamido)benzoic...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding to low affinity site of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50209511(5-cyano-2-(2-(3-(2-methoxyethoxy)propylthio)nicoti...)
Affinity DataKd:  700nMAssay Description:Binding affinity to human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219742(5-fluoro-2-(3-(morpholinosulfonyl)benzamido)benzoi...)
Affinity DataKd:  6.60E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219743(2-(3-(morpholinosulfonyl)benzamido)-5-nitrobenzoic...)
Affinity DataKd:  4.40E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50219744(2-(3-(morpholinosulfonyl)benzamido)benzoic acid | ...)
Affinity DataKd:  6.00E+3nMAssay Description:Displacement of fluorescent dansyl sarcosine from human serum albumin site II on subdomain IIIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed