Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from rat BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from mouse BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]D-Tyr6-betaAla11-Phe13-Nle14-bombesin from human BRS-3 expressed in NFAT-CHO cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair
TargetAmiloride-sensitive sodium channel subunit alpha(Homo sapiens (Human))
Parion Sciences
Curated by ChEMBL
Parion Sciences
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assayMore data for this Ligand-Target Pair