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Found 3817 with Last Name = 'swinger' and Initial = 'kk'
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50365695(CHEMBL1958408)
Affinity DataKi:  0.280nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426461(CHEMBL2322677)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426464(CHEMBL2322674)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426467(CHEMBL2322683)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426468(CHEMBL2322682)
Affinity DataKi:  3.20nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426466(CHEMBL2322684)
Affinity DataKi:  3.40nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426463(CHEMBL2322675)
Affinity DataKi:  5.5nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426465(CHEMBL2322673)
Affinity DataKi:  7.70nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426472(CHEMBL2322678)
Affinity DataKi:  8.70nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426471(CHEMBL2322679)
Affinity DataKi:  13nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426470(CHEMBL2322680)
Affinity DataKi:  15nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426469(CHEMBL2322681)
Affinity DataKi:  27nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426461(CHEMBL2322677)
Affinity DataKi:  58nMAssay Description:Inhibition of human recombinant GSK3betaMore data for this Ligand-Target Pair
TargetCell division cycle 7-related protein kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50426462(CHEMBL2322676)
Affinity DataKi:  67nMAssay Description:Inhibition of human Cdc7 using biotin-C6linker-TPSDSLIYDDGLS as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344200((2R)-1-[3-{[6-(4-acetylpiperazin-1-yl)-2-ethoxypyr...)
Affinity DataIC50:  1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344204((2R)-2-[3-{[6-(4-acetylpiperazin-1-yl)-2-ethoxypyr...)
Affinity DataIC50:  1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344248(N-{6-[(3S)-4-acetyl-3-(methoxymethyl)piperazin-1-y...)
Affinity DataIC50:  1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 8(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095355(CHEMBL3589029)
Affinity DataIC50:  2nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT8 expressed in Escherichia coli (BL21(DE3) pre-incubated for 30 mins before addition of a [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095436(CHEMBL3589043)
Affinity DataIC50:  2nMAssay Description:Inhibition of FLAG and hexa-histidine tagged full-length human PRMT6 expressed in HEK293F cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095355(CHEMBL3589029)
Affinity DataIC50:  2nMAssay Description:Inhibition of FLAG and hexa-histidine tagged full-length human PRMT6 expressed in HEK293F cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344282(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  2.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344241(N-{6-[(2S)-2-(hydroxymethyl)-4-(morpholin-4-ylcarb...)
Affinity DataIC50:  2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344245(N-{6-[(2R)-4-acetyl-2-(hydroxymethyl)piperazin-1-y...)
Affinity DataIC50:  2.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344277(N-[6-(4-acetylpiperazin-1-yl)-2-methoxypyridin-3-y...)
Affinity DataIC50:  2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095438(CHEMBL3589042)
Affinity DataIC50:  3nMAssay Description:Inhibition of FLAG and hexa-histidine tagged full-length human PRMT6 expressed in HEK293F cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344224(N-{6-[4-(N′-cyano-N-methylcarbamimidoyl)pipe...)
Affinity DataIC50:  3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344222(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  3.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344239(N-{6-[(3S)-4-acetyl-3-(hydroxymethyl)piperazin-1-y...)
Affinity DataIC50:  3.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344205(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  3.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344279(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  3.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344290(N-[6-(1-acetylpiperidin-4-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  3.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344217(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344240(N-{6-[(2S)-4-acetyl-2-(hydroxymethyl)piperazin-1-y...)
Affinity DataIC50:  3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095354(CHEMBL3589030)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095432(CHEMBL3589026)
Affinity DataIC50:  4nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344264(N-[4-(4-acetylpiperazin-1-yl)-2-methoxyphenyl]-6,6...)
Affinity DataIC50:  4.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50315895(CHEMBL1090357 | N-(3-(5-(2-(4-(2-(dimethylamino)et...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344201(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  4.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344195(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344196(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344281(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344289(N-{6-(4-acetylpiperazin-1-yl)-2-[(1-oxidothietan-3...)
Affinity DataIC50:  4.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344203(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  4.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50315905(CHEMBL1090350 | N-(3-(5-(2-(4-morpholinophenylamin...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of ErbB2 by time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344285(N-[6-(4-acetylpiperazin-1-yl)-2-(oxetan-3-yloxy)py...)
Affinity DataIC50:  4.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095353(CHEMBL3589031)
Affinity DataIC50:  5nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095356(CHEMBL3589028)
Affinity DataIC50:  5nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 6(Homo sapiens (Human))
Epizyme

Curated by ChEMBL
LigandPNGBDBM50095435(CHEMBL3590417)
Affinity DataIC50:  5nMAssay Description:Inhibition of FLAG and hexa-histidine tagged full-length human PRMT6 expressed in HEK293F cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344115(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  5.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344280(N-[6-(4-acetylpiperazin-1-yl)-2-ethoxypyridin-3-yl...)
Affinity DataIC50:  5.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 3817 total ) | Next | Last >>
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