TargetCytochrome P450 2C9(Homo sapiens (Human))
University Of North Carolina At Greensboro
Curated by ChEMBL
University Of North Carolina At Greensboro
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of CYP2C9 in pooled human liver microsomes assessed as reduction in enzyme-mediated (S)-warfarin 7-hydroxylation by HPLC/MS-MS methodMore data for this Ligand-Target Pair