TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
National Institutes Of Health
Curated by ChEMBL
National Institutes Of Health
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Affinity for the Corticotropin releasing factor receptor 1 (CRHR1) was determined in rat brainMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
National Institute Of Biomedical Imaging And Bioengineering
Curated by ChEMBL
National Institute Of Biomedical Imaging And Bioengineering
Curated by ChEMBL
Affinity DataIC50: 27.4nMAssay Description:Antagonist activity at CXCR4 in human Jurkat cells assessed as inhibition of SDF1-induced cell migrationMore data for this Ligand-Target Pair
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
National Institute Of Biomedical Imaging And Bioengineering
Curated by ChEMBL
National Institute Of Biomedical Imaging And Bioengineering
Curated by ChEMBL
Affinity DataIC50: 1.52E+4nMAssay Description:Displacement of [125I]SDF1alpha from CXCR4 in human HL60 cellsMore data for this Ligand-Target Pair