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Found 44 with Last Name = 'thomas' and Initial = 'be'
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125708(1-(3,5-Dichloro-phenyl)-3-{3-[3-(3,5-dichloro-phen...)
Affinity DataIC50:  480nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125717(1-{2,4-Dibromo-5-[3-(4-iodo-phenyl)-ureido]-phenyl...)
Affinity DataIC50:  590nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125729(3,5-Dichloro-N-{3-[3-(2,4-dibromo-phenyl)-ureido]-...)
Affinity DataIC50:  620nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125714(3,5-Dichloro-N-{3-[3-(3,5-dichloro-phenyl)-ureido]...)
Affinity DataIC50:  690nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125731(3,5-Dichloro-N-[3-(3,3-diphenyl-propionylamino)-ph...)
Affinity DataIC50:  870nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125720(3,5-Dichloro-N-[3-(2-naphthalen-2-yl-acetylamino)-...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125716(3,5-dichloro-N-{3-[(3,5-dichlorobenzoyl)amino]phen...)
Affinity DataIC50:  930nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125706(3,5-Dichloro-N-{3-[3-(4-trifluoromethyl-phenyl)-ur...)
Affinity DataIC50:  940nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125718(1,3-di(5-chloro-2-methylsulfonylphenylcarboxamido)...)
Affinity DataIC50:  1.02E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125721(3,5-Dichloro-N-[3-(2-naphthalen-1-yl-acetylamino)-...)
Affinity DataIC50:  1.12E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125715(3,5-Dichloro-N-[3-(3-phenyl-ureido)-phenyl]-benzam...)
Affinity DataIC50:  1.18E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125719(3,5-Dichloro-N-{3-[3-(2-ethyl-phenyl)-ureido]-phen...)
Affinity DataIC50:  1.41E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125722(1-Naphthalen-1-ylmethyl-3-[3-(3-naphthalen-1-ylmet...)
Affinity DataIC50:  1.92E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125724(3,5-Dichloro-N-{3-[3-(2-methyl-benzyl)-ureido]-phe...)
Affinity DataIC50:  2.12E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125709(1-{2,4-Dibromo-5-[3-(4-dimethylamino-phenyl)-ureid...)
Affinity DataIC50:  2.90E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125732(1-(3,5-Dichloro-phenyl)-3-{3-[3-(3,5-dichloro-phen...)
Affinity DataIC50:  2.95E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125713(CHEMBL276713 | N-[3-(3-Benzyl-ureido)-phenyl]-3,5-...)
Affinity DataIC50:  3.35E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125728(CHEMBL13550 | N-(3,5-dichlorophenyl)-N'-{3-[({[(3,...)
Affinity DataIC50:  3.95E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125707(1-Isoxazol-3-yl-3-[3-(3-isoxazol-3-yl-ureido)-phen...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125727(1-(3,5-Dichloro-phenyl)-3-{3-[3-(3,5-dichloro-phen...)
Affinity DataIC50:  4.20E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125710(1-Naphthalen-1-yl-3-[3-(3-naphthalen-1-yl-ureido)-...)
Affinity DataIC50:  4.55E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125712(1-(2,2-Diphenyl-ethyl)-3-{3-[3-(2,2-diphenyl-ethyl...)
Affinity DataIC50:  4.85E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125723(1-(2,4-Dibromo-phenyl)-3-{3-[3-(2,4-dibromo-phenyl...)
Affinity DataIC50:  5.09E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125725(1,1'-(4,6-dibromo-1,3-phenylene)bis(3-(2-carbamoyl...)
Affinity DataIC50:  5.90E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125730(1-(2,4-Dibromo-phenyl)-3-{3-[3-(2,4-dibromo-phenyl...)
Affinity DataIC50:  6.20E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125711(1-(2,4-Dimethyl-phenyl)-3-{3-[3-(2,4-dimethyl-phen...)
Affinity DataIC50:  8.50E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Rattus norvegicus)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50125726(1-(3-Methoxy-phenyl)-3-{3-[3-(3-methoxy-phenyl)-ur...)
Affinity DataIC50:  9.50E+3nMAssay Description:In vitro inhibition of the rotamase activity of cyclophilin A (CyPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50450369(SIALYL LEWIS X | Sialyl LeX | Sialyl lewis-x | sLe...)
Affinity DataIC50:  3.00E+5nMAssay Description:In vitro inhibitory activity against binding of Selectin E to human recombinant AGP (alpha-1 acid glycoprotein) containing sLex derivativeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096284(2-{2-[6-(4-Benzyl-4-hydroxy-piperidin-1-ylmethyl)-...)
Affinity DataIC50:  1.60E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin glycoprotein ligand 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50111451(2-[2-(3,4,5-Trihydroxy-6-{[2-(1-phenyl-ethylcarbam...)
Affinity DataIC50:  2.50E+6nMAssay Description:Ability to inhibit the binding of P-selectin glycoprotein ligand 1 (PSGL-1) fusion protein to immobilized soluble P-selectin in a P-selectin assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096291(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  3.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1-acid glycoprotein 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50111451(2-[2-(3,4,5-Trihydroxy-6-{[2-(1-phenyl-ethylcarbam...)
Affinity DataIC50:  5.00E+6nMAssay Description:Ability to inhibit the binding of E-selectin to human recombinant AGP (alpha-1 acid glycoprotein) in a E-selectin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096293(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  6.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096287(5-({6-[(1,3-Dicarboxy-propylcarbamoyl)-methyl]-3,4...)
Affinity DataIC50:  6.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096290(2-(2-{6-[(1-Carbamoyl-2-phenyl-ethylamino)-methyl]...)
Affinity DataIC50:  6.70E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096289(2-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-...)
Affinity DataIC50:  7.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096292(6-Amino-2-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tet...)
Affinity DataIC50:  7.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096286(2-[2-(3,4,5-Trihydroxy-6-{[methyl-(3-methyl-cycloh...)
Affinity DataIC50:  8.00E+6nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1-acid glycoprotein 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50111453((4R,5S)-2-{[(3S,4S,5S)-2-{[(2S,3S)-5-acetamido-6-h...)
Affinity DataIC50:  8.00E+6nMAssay Description:Ability to inhibit the binding of E-selectin to human recombinant AGP (alpha-1 acid glycoprotein) in a E-selectin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096294(4-Carbamoyl-2-[2-(3,4,5-trihydroxy-6-hydroxymethyl...)
Affinity DataIC50: >1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin(Homo sapiens (Human))
Wyeth

Curated by ChEMBL
LigandPNGBDBM50169053((3R,5R)-3,4,5-Trihydroxy-1-(2'-trifluoromethyl-bip...)
Affinity DataIC50:  1.00E+7nMAssay Description:Inhibitory concentration against selectin P in Biacore assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096285(3-{4-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahyd...)
Affinity DataIC50:  1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE-selectin(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50096288(4-{4-[2-(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahyd...)
Affinity DataIC50: >1.00E+7nMAssay Description:In vitro inhibitory activity against Selectin E binding to human recombinant AGP (alpha-1 acid glycoprotein)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP-selectin glycoprotein ligand 1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50111452((4R,5S)-5-[({[6-({[(1S)-1,3-dicarboxypropyl]carbam...)
Affinity DataIC50:  2.50E+8nMAssay Description:Ability to inhibit the binding of P-selectin glycoprotein ligand 1 (PSGL-1) fusion protein to immobilized soluble P-selectin in a P-selectin assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed