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Found 14 with Last Name = 'trantolo' and Initial = 'dj'
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022163(6-(Indan-5-ylamino)-1H-pyrimidine-2,4-dione | CHEM...)
Affinity DataKi:  400nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the presence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022167(2-Amino-6-(indan-5-ylamino)-3H-pyrimidin-4-one | C...)
Affinity DataKi:  2.00E+3nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the presence of dATP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022154(6-Benzylamino-1H-pyrimidine-2,4-dione | CHEMBL8648...)
Affinity DataKi:  7.50E+3nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the presence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022146(6-Benzylamino-5-bromo-1H-pyrimidine-2,4-dione | CH...)
Affinity DataKi:  9.00E+3nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022155(6-Benzylamino-5-iodo-1H-pyrimidine-2,4-dione | CHE...)
Affinity DataKi:  9.00E+3nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022142(5-Bromo-6-p-tolylamino-1H-pyrimidine-2,4-dione | C...)
Affinity DataKi:  1.40E+4nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022161(6-p-Tolylamino-1H-pyrimidine-2,4-dione | CHEMBL573...)
Affinity DataKi:  1.70E+4nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the presence of dATP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022150(CHEMBL158113 | N*4*-Benzyl-6-chloro-pyrimidine-2,4...)
Affinity DataKi:  1.70E+4nMAssay Description:Compound was tested for its inhibitory activity against Bacillus subtilis DNA topoisomerase III using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022149(6-Benzylamino-1H-[1,3,5]triazine-2,4-dione | CHEMB...)
Affinity DataKi:  2.00E+4nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022168(2-Amino-6-benzylamino-3H-pyrimidin-4-one | CHEMBL3...)
Affinity DataKi:  3.30E+4nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the presence of dATP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022148(6-p-Tolylamino-1H-[1,3,5]triazine-2,4-dione | CHEM...)
Affinity DataKi:  7.00E+4nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022138(6-Benzylamino-5-methyl-1H-pyrimidine-2,4-dione | C...)
Affinity DataKi:  4.36E+5nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dCTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022160(5-Methyl-6-p-tolylamino-1H-pyrimidine-2,4-dione | ...)
Affinity DataKi:  1.58E+6nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 3(Bacillus subtilis)
TBA

Curated by ChEMBL
LigandPNGBDBM50022145(6-Benzylamino-5-ethyl-1H-pyrimidine-2,4-dione | CH...)
Affinity DataKi:  2.82E+6nMAssay Description:Concentration producing 50% inhibition of Bacillus subtilis DNA topoisomerase III in the absence of dGTP using DNA Polymerase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed