Affinity DataKi: 0.800nMAssay Description:Inhibition of caspase 1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of caspase 1 (unknown origin)More data for this Ligand-Target Pair
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of telomerase activity in human M14 cells using biotin-labeled TeloTAGGG as primer preincubated for 48 hrs followed by primer addition mea...More data for this Ligand-Target Pair
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of telomerase activity in human HT-29 cells using biotin-labeled TeloTAGGG as primer preincubated for 48 hrs followed by primer addition m...More data for this Ligand-Target Pair
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of telomerase activity in human MCF7 cells using biotin-labeled TeloTAGGG as primer preincubated for 48 hrs followed by primer addition me...More data for this Ligand-Target Pair
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Istituto Di Farmacologia Traslazionale
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of telomerase activity in human H125 cells using biotin-labeled TeloTAGGG as primer preincubated for 48 hrs followed by primer addition me...More data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.26E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.14E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.35E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 7.78E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 7.94E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 9.41E+4nMAssay Description:Inhibition of caspase 1 (unknown origin) using YVAD-AFC as substrate by fluorescence analysisMore data for this Ligand-Target Pair