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Found 4892 with Last Name = 'urbano' and Initial = 'm'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  0.0200nMAssay Description:Antagonist activity at kappa opioid receptor in guinea pig caudate assessed as inhibition of U69593-stimulated [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357453(CHEMBL1917719)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357441(CHEMBL1917705)
Affinity DataKi:  0.860nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357440(CHEMBL1917704)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198054((3-biphenyl-4-yl-butyl)-dimethyl-amine | CHEMBL224...)
Affinity DataKi:  1.02nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357430(CHEMBL1917711)
Affinity DataKi:  1.07nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50350976(CHEMBL1818341)
Affinity DataKi:  1.20nMAssay Description:Antagonist activity at human cloned kappa opioid receptor expressed in CHO cells assessed as inhibition of U69593-stimulated [35S]-GTP[gammaS] bindin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310078((R/S)-1-(3-(6-Methoxynaphthalen-2-yl)butyl)piperid...)
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198061((E)-N,N-dimethyl-3-(biphen-4-yl)but-2-en-1-ylamine...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198061((E)-N,N-dimethyl-3-(biphen-4-yl)but-2-en-1-ylamine...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50531908(Btrx-335140 | CYM-53093 | US10676469, Compound 142...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]diprenorphine from human KORMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50012152(CHEMBL3264441)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]diprenorphine from kappa opioid receptor (unknown origin) expressed in CHO cells membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198064(CHEMBL224855 | N,N-dimethyl-3-(naphthalen-2-yl)but...)
Affinity DataKi:  1.95nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50130563((3R)-7-Hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphe...)
Affinity DataKi:  2.20nMAssay Description:Antagonist activity at mu opioid receptor in guinea pig caudate assessed as inhibition of DAMGO-stimulated [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198055((R/S)-3-(6-Methoxynaphthalen-2-yl)-N,N-dimethylbut...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310077((R/S)-N-Benzyl-3-(6-methoxynaphthalen-2-yl)-N-meth...)
Affinity DataKi:  2.31nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310074((R/S)-4-(benzyl(methyl)amino)-2-(biphenyl-4-yl)but...)
Affinity DataKi:  2.38nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198062((R/S)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbutan-1-a...)
Affinity DataKi:  3.59nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357431(CHEMBL1917712)
Affinity DataKi:  4.14nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198065(4(E)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbut-2-en-1...)
Affinity DataKi:  4.17nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310076((E)-1-(3-(6-Methoxynaphthalen-2-yl)but-2-enyl)pipe...)
Affinity DataKi:  4.41nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357429(CHEMBL1917702)
Affinity DataKi:  5.25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198063(CHEMBL387955 | N-benzyl-N-methyl-3-(naphthalen-2-y...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198062((R/S)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbutan-1-a...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310072((R/S)-4-(Benzyl(methyl)amino)-2-(6-methoxynaphthal...)
Affinity DataKi:  6.04nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198065(4(E)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbut-2-en-1...)
Affinity DataKi:  6.32nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198065(4(E)-N-Benzyl-3-(biphenyl-4-yl)-N-methylbut-2-en-1...)
Affinity DataKi:  6.32nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50012151(CHEMBL3264440)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]diprenorphine from mu opioid receptor (unknown origin) expressed in CHO cells membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357446(CHEMBL1917710)
Affinity DataKi:  7.02nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357447(CHEMBL1917713)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198058((E)-N-benzyl-N-methyl-3-(naphthalen-2-yl)but-2-en-...)
Affinity DataKi:  7.88nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198058((E)-N-benzyl-N-methyl-3-(naphthalen-2-yl)but-2-en-...)
Affinity DataKi:  7.88nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357448(CHEMBL1917714)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50350976(CHEMBL1818341)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human cloned mu opioid receptor expressed in CHO cells assessed as inhibition of DAMGO-stimulated [35S]-GTP[gammaS] bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357432(CHEMBL1917703)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310073((R/S)-2-(6-Methoxynaphthalen-2-yl)-4-(piperidin-1-...)
Affinity DataKi:  10.4nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357449(CHEMBL1917715)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50310075((E)-N-Benzyl-3-(6-methoxynaphthalen-2-yl)-N-methyl...)
Affinity DataKi:  13.7nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357443(CHEMBL1917707)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198055((R/S)-3-(6-Methoxynaphthalen-2-yl)-N,N-dimethylbut...)
Affinity DataKi:  14.4nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 opioid receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198067((R/S)-N,N-dimethyl-3-(6-hydroxy-naphthalen-2-yl)bu...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198068((E)-N,N-dimethyl-3-(naphthalen-2-yl)but-2-en-1-ami...)
Affinity DataKi:  19.8nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198068((E)-N,N-dimethyl-3-(naphthalen-2-yl)but-2-en-1-ami...)
Affinity DataKi:  19.8nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50248984(CHEMBL473989 | N-Benzyl-3-[1-(4-fluorophenyl)-1H-i...)
Affinity DataKi:  20.8nMAssay Description:Displacement of [3H] (+)-pentazocine from sigma 1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50264571(CHEMBL523473 | N-(2,4-Dimethylbenzyl)-4-[1-(4-fluo...)
Affinity DataKi:  20.8nMAssay Description:Displacement of [3H] (+)-pentazocine from sigma 1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198066((E)-3-(6-Methoxynaphthalen-2-yl)-N,N-dimethylbut-2...)
Affinity DataKi:  21.4nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50357445(CHEMBL1917709)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50012151(CHEMBL3264440)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]diprenorphine from kappa opioid receptor (unknown origin) expressed in CHO cells membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL
LigandPNGBDBM50198057((R/S)-4-(dimethylamino)-2-(naphthalen-2-yl)butan-2...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50012152(CHEMBL3264441)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]diprenorphine from mu opioid receptor (unknown origin) expressed in CHO cells membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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