Affinity DataKi: 0.310nMAssay Description:Mixed-type inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradish peroxidase-A...More data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Non-competitive inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in...More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
Affinity DataKi: 0.790nMAssay Description:Competitive inhibition of human microsomal MAO-B expressed in recombinant baculovirus infected insect BTI-TN-5B1-4 cells assessed as reduction in H2O...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Noncompetitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate as...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as substrate assessed as decre...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Compound was measured for the inhibition of [3H]-8-OH-DPAT binding to rat hippocampus membrane (5-HT1A receptor)More data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Non-competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradish peroxid...More data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Porto
Curated by ChEMBL
University Of Porto
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of electric eel AChE assessed as inhibition constant using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Compound was measured for the binding affinity in homogenated mouse fibroblast (LTK) cells transfected with human Dopamine receptor D2A using [3H]-ra...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Tight-binding competitive inhibition of recombinant human MAO-B expressed in Pichia pastoris using benzylamine as substrate by fluorimetric horseradi...More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOA expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Compound was measured for the binding affinity in chinese hamster ovary (CHO) cells transfected with human Dopamine receptor D3 using [3H]-raclopride...More data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Mixed type inhibition of human AChE using acetylthiocholine iodide as substrate pretreated for 5 mins followed by substrate addition measured after 5...More data for this Ligand-Target Pair
Affinity DataKi: 258nMAssay Description:Displacement of [3H]HEMADO from human adenosine receptor A3 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 324nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Affinity DataKi: 478nMAssay Description:Reversible competitive inhibition of human recombinant microsomal MAOB expressed in baculovirus infected BTI-TN-5B1- 4 cells using p-tyramine as subs...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 537nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 562nMAssay Description:Binding affinity towards Dopamine receptor D2 in rat frontal striatum using [3H]spiperoneMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 933nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+3nMAssay Description:Displacement of [3H]NECA from human adenosine receptor A2A expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 1.95E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Santiago
Curated by ChEMBL
University Of Santiago
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor using [3H]ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine receptor A1 expressed in CHO cell membranes by radioligand competition assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.89E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair