TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase in membrane vesicle from BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of ATPase in membrane vesicle from BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Hungarian Academy Of Sciences
Curated by ChEMBL
Hungarian Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:TP_TRANSPORTER: efflux of Hoechst33342 in BCRP-expressing Sf9 cellsMore data for this Ligand-Target Pair