Affinity DataKi: 180nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 3.98E+4nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+4nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 4.17E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 9.05E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of [14C]-Gly-Sar transport by hPEPT1 in Caco-2 cell monolayersMore data for this Ligand-Target Pair
Affinity DataIC50: 4.05E+4nMAssay Description:Concentration required to inhibit the maximum [14C]-Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of [14C]-Gly-Sar transport by hPEPT1 in Caco-2 cell monolayersMore data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+5nMAssay Description:Inhibition of [14C]-Gly-Sar transport by hPEPT1 in Caco-2 cell monolayersMore data for this Ligand-Target Pair
Affinity DataIC50: 4.22E+5nMAssay Description:Inhibition of [14C]-Gly-Sar transport by hPEPT1 in Caco-2 cell monolayersMore data for this Ligand-Target Pair
Affinity DataIC50: 9.15E+5nMAssay Description:Inhibition of [14C]-Gly-Sar transport by hPEPT1 in Caco-2 cell monolayersMore data for this Ligand-Target Pair
Affinity DataEC50: 1.48E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 7.24E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 661nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 257nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 562nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 5.37E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.95E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.86E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 3.55E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 3.63E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 776nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 676nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 2.88E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 470nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 780nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 5.40E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 660nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 468nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 680nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 7.20E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair