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Found 41 with Last Name = 'valadés' and Initial = 'ea'
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349983(CHEMBL1812596)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252920((S)-1-[2'-Amino-2'-carboxyethyl]-5,7-dihydrothieno...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252922((S)-1-(2'-Amino-2'-carboxyethyl)thieno[3,2-d]pyrim...)
Affinity DataKi:  5.29nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349981(CHEMBL1812598)
Affinity DataKi:  5.89nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50207593((S)-1-(2-AMINO-2-CARBOXYETHYL)-3(2-CARBOXYTHIOPHEN...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252920((S)-1-[2'-Amino-2'-carboxyethyl]-5,7-dihydrothieno...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252922((S)-1-(2'-Amino-2'-carboxyethyl)thieno[3,2-d]pyrim...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349980(CHEMBL1738726)
Affinity DataKi:  157nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349983(CHEMBL1812596)
Affinity DataKi:  465nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349981(CHEMBL1812598)
Affinity DataKi:  503nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349979(CHEMBL1812599)
Affinity DataKi:  567nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349983(CHEMBL1812596)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252920((S)-1-[2'-Amino-2'-carboxyethyl]-5,7-dihydrothieno...)
Affinity DataKi:  3.25E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252922((S)-1-(2'-Amino-2'-carboxyethyl)thieno[3,2-d]pyrim...)
Affinity DataKi:  3.65E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349982(CHEMBL1812597)
Affinity DataKi:  3.67E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349981(CHEMBL1812598)
Affinity DataKi:  4.75E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi:  5.09E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349980(CHEMBL1738726)
Affinity DataKi:  7.45E+3nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349977(CHEMBL1812601)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(RAT)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349978(CHEMBL1812600)
Affinity DataKi:  1.51E+4nMAssay Description:Displacement of [3H]SYM2081 from rat GluK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349979(CHEMBL1812599)
Affinity DataKi:  5.38E+4nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349982(CHEMBL1812597)
Affinity DataKi:  7.23E+4nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349980(CHEMBL1738726)
Affinity DataKi:  7.29E+4nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349980(CHEMBL1738726)
Affinity DataKi:  9.90E+4nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349979(CHEMBL1812599)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349977(CHEMBL1812601)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349983(CHEMBL1812596)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349982(CHEMBL1812597)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349979(CHEMBL1812599)
Affinity DataKi:  1.08E+5nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349977(CHEMBL1812601)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349978(CHEMBL1812600)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349978(CHEMBL1812600)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349977(CHEMBL1812601)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK3 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349981(CHEMBL1812598)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349982(CHEMBL1812597)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50349978(CHEMBL1812600)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]AMPA from rat GluA2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50107595((S)-1-(2-Amino-2-carboxyethyl)-6,7-dihydro-1H-cycl...)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252920((S)-1-[2'-Amino-2'-carboxyethyl]-5,7-dihydrothieno...)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252922((S)-1-(2'-Amino-2'-carboxyethyl)thieno[3,2-d]pyrim...)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]SYM2081 from rat GluK2 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed