Affinity DataKi: 93nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.42E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.64E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 5.62E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair