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Found 62 with Last Name = 'van lint' and Initial = 'j'
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  3.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  4.83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  8.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  11.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  24.6nMMore data for this Ligand-Target Pair
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  26.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  28.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  43.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  48.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  146nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  224nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565693(CHEMBL4515390)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565693(CHEMBL4515390)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565693(CHEMBL4515390)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565690(CHEMBL4787572)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565690(CHEMBL4787572)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565690(CHEMBL4787572)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565692(CHEMBL4790321)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM416549(US10307425, Example 15 | US10632122, Example 15)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565692(CHEMBL4790321)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565691(CHEMBL4776166)
Affinity DataIC50:  55nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D1(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565691(CHEMBL4776166)
Affinity DataIC50:  64nMAssay Description:Inhibition of recombinant FLAG-tagged PKD1 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565692(CHEMBL4790321)
Affinity DataIC50:  76nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D3(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565691(CHEMBL4776166)
Affinity DataIC50:  78nMAssay Description:Inhibition of recombinant FLAG-tagged PKD3 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50565687(CHEMBL4779081)
Affinity DataIC50:  94nMAssay Description:Inhibition of recombinant FLAG-tagged PKD2 (unknown origin) expressed in HEK293T cells using Syntide-2 as substrate measured after 15 mins by ADP-Glo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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