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Found 39 with Last Name = 'vancraeynest' and Initial = 'c'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human DYRK1A kinase expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019771(CHEMBL3286602)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019769(CHEMBL3286600)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019768(CHEMBL3286599)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019762(CHEMBL3286595)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019770(CHEMBL3286601)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019763(CHEMBL3286596)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019765(CHEMBL3286597)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333423(7-(Pyridin-3-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395379(CHEMBL2164712 | US9168247, CV12)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019783(CHEMBL3286612)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019764(CHEMBL1528603)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333416(7-(2-Methoxyethoxy)-1-methyl-beta-carboline | CHEM...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395380(CHEMBL2164709 | US9168247, JR84)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019784(CHEMBL3286613)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019778(CHEMBL3286607)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019787(CHEMBL3286615)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019776(CHEMBL3286606)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019766(CHEMBL3286598)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395378(CHEMBL2164696 | US9168247, CV24)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019782(CHEMBL3286611)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019772(CHEMBL3286603)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019767(CHEMBL1542642)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019786(CHEMBL3286614)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019788(CHEMBL3286616)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019789(CHEMBL3286617)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019790(CHEMBL3286618)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019791(CHEMBL3286619)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019761(CHEMBL3286594)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019760(CHEMBL1521164)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019759(CHEMBL3286593)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019781(CHEMBL3286610)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019780(CHEMBL3286609)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019779(CHEMBL3286608)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019773(CHEMBL3286604)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019774(CHEMBL444521)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50019775(CHEMBL3286605)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
University Of Namur (Unamur)

Curated by ChEMBL
LigandPNGBDBM50241727((S)-2-amino-3-(1-methyl-1H-indol-3-yl)propanoic ac...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant N-terminal His-tagged human IDO (Ala2 to Gly403) overexpressed in Escherichia coli BL21 AI using L-tryptophan as substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed