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Found 96 with Last Name = 'vandenberg' and Initial = 'rj'
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | 3-aminopropylphos...)
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM24185((3-aminopropyl)(methyl)phosphinic acid | 3-Apmpa |...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataKi:  280nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi:  650nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM24185((3-aminopropyl)(methyl)phosphinic acid | 3-Apmpa |...)
Affinity DataKi:  750nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM24184((3-aminopropyl)phosphinic acid | 3-aminopropylphos...)
Affinity DataKi:  2.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataKi:  4.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi:  5.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataKi:  6.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataKi:  7.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032982((3-Amino-propyl)-butyl-phosphinic acid | 3-aminopr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032982((3-Amino-propyl)-butyl-phosphinic acid | 3-aminopr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032962(((Z)-3-Amino-propenyl)-phosphinic acid | CGP38593 ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(((Z)-3-Amino-propenyl)-methyl-phosphinic acid | 3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(4-Benzyloxy-N-(1-dimethylamino-cyclopentylmethyl)-...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50102692(4-Benzyloxy-N-(1-dimethylamino-cyclopentylmethyl)-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human GlyT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537022(CHEMBL4587165)
Affinity DataIC50:  26nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537040(CHEMBL4515597)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537034(CHEMBL4572247)
Affinity DataIC50:  32nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537033(CHEMBL4535356)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537044(CHEMBL4562565)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537043(CHEMBL4227139)
Affinity DataIC50:  55nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537049(CHEMBL4527071)
Affinity DataIC50:  65nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537023(CHEMBL4542099)
Affinity DataIC50:  69nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537054(CHEMBL4549008)
Affinity DataIC50:  91nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50256745((2S)-2-amino-3-((2-(benzyloxy)phenyl)(3-fluorophen...)
Affinity DataIC50:  100nMAssay Description:Inhibition of full length human GlyT2 expressed in FreeStyle 293-F suspension cells incubated for 30 mins before [3H]glycine addition and measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50023924(CHEMBL3325507)
Affinity DataIC50:  105nMAssay Description:Reversible inhibition of recombinant human GlyT2 expressed in HEK293 cells assessed as reduction in [3H]-glycine uptake after 2 hrs by top count assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537031(CHEMBL4540633)
Affinity DataIC50:  130nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537017(CHEMBL4228560)
Affinity DataIC50:  143nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537029(CHEMBL4592570)
Affinity DataIC50:  151nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537045(CHEMBL4562110)
Affinity DataIC50:  152nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537035(CHEMBL4549529)
Affinity DataIC50:  182nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537028(CHEMBL4228763)
Affinity DataIC50:  214nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537048(CHEMBL4576431)
Affinity DataIC50:  259nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537019(CHEMBL4526987)
Affinity DataIC50:  259nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537032(CHEMBL4559571)
Affinity DataIC50:  313nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537046(CHEMBL4531406)
Affinity DataIC50:  340nMAssay Description:Reversible non-competitive inhibition of human GlyT2a expressed in Xenopus laevis oocytes by two-electrode voltage clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537041(CHEMBL4515758)
Affinity DataIC50:  496nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537018(CHEBI:73723 | Oleoyl Glycine)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537018(CHEBI:73723 | Oleoyl Glycine)
Affinity DataIC50:  500nMAssay Description:Reversible non-competitive inhibition of human GlyT2a expressed in Xenopus laevis oocytes by two-electrode voltage clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537036(CHEMBL4559157)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537024(CHEBI:17490 | CHEMBL3392050)
Affinity DataIC50:  600nMAssay Description:Reversible non-competitive inhibition of human GlyT2a expressed in Xenopus laevis oocytes by two-electrode voltage clamp electrophysiologyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537042(CHEMBL4526841)
Affinity DataIC50:  613nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537025(CHEMBL4545242)
Affinity DataIC50:  865nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537047(CHEMBL4543598)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 2(Homo sapiens (Human))
University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50537038(CHEMBL4516669)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of recombinant human GlyT2a expressed in Xenopus laevis oocytes assessed as reduction in channel current by two-electrode voltage clamp el...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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