Compile Data Set for Download or QSAR
maximum 50k data
Found 57 with Last Name = 'vanderesse' and Initial = 'r'
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185622(Apam-YET | CHEMBL210325)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185622(Apam-YET | CHEMBL210325)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi:  1.50E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185649((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185650(CHEMBL209568 | Pam-YET)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185650(CHEMBL209568 | Pam-YET)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185626((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185641(CHEMBL209984 | Pam-YNT)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185621((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185642((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185637((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185640((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185648((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  4.30E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185638((S)-2-{(S)-4-Carboxy-2-[(S)-2-hexanoylamino-3-(4-h...)
Affinity DataKi:  5.90E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi:  6.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185619((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185632((S)-2-{(S)-4-carboxy-2-[(S)-2-decanoylamino-3-(4-h...)
Affinity DataKi:  7.20E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185624((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185627((S)-2-{(S)-4-Carboxy-2-[(S)-3-(4-hydroxy-phenyl)-2...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185651((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185645((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185648((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185647((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185638((S)-2-{(S)-4-Carboxy-2-[(S)-2-hexanoylamino-3-(4-h...)
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)
Affinity DataKi:  8.10E+4nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185620(CHEMBL378655 | TVTFKF)
Affinity DataKi:  1.39E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185620(CHEMBL378655 | TVTFKF)
Affinity DataKi:  1.48E+5nMAssay Description:Inhibition of post acid activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185629(CHEMBL277277 | TITYKF)
Affinity DataKi:  1.51E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-6(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185629(CHEMBL277277 | TITYKF)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of post acid activity of yeast 20S proteasome at 625 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)
Affinity DataKi:  3.15E+5nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185636(CHEMBL210501 | TVTYKL)
Affinity DataKi:  5.45E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185639(CHEMBL378045 | TITYDL)
Affinity DataKi:  6.19E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185623(CHEMBL426505 | TVSYKF)
Affinity DataKi: >6.25E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185631(CHEMBL426136 | TISYDY)
Affinity DataKi: >6.25E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Saccharomyces cerevisiae)
Cnrs-Université

Curated by ChEMBL
LigandPNGBDBM50185634(CHEMBL378002 | TITFDY)
Affinity DataKi: >6.25E+5nMAssay Description:Inhibition of chymotrypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 57 total ) | Next | Last >>
Jump to: