Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 135nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from Sprague-Dawley rat cerebral cortex H3 receptor measured after 30 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 454nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Displacement of [3H]methyl- N-alpha methylhistamine dihydrochloride from human recombinant H3 receptor expressed in CHOK1 cells measured after 30 min...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Chemical Works Of Gedeon Richter
Curated by ChEMBL
Affinity DataKi: 700nMAssay Description:Displacement of [3H]quinuclidinyl benzilate from Wistar rat cortex muscarinic acetylcholine receptor by liquid scintillation counter methodMore data for this Ligand-Target Pair