Affinity DataIC50: 7.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 118nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 134nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 163nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 181nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 299nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 312nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 524nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using receptor binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 2.33E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Activation of PXR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Gedeon Richter
Curated by ChEMBL
Gedeon Richter
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human ERG by patch clamp electrophysiology assayMore data for this Ligand-Target Pair