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Found 705 with Last Name = 'vargas' and Initial = 'h'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108699(1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfony...)
Affinity DataKi:  0.420nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84445(Isoindoline, 12)
Affinity DataKi:  0.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  0.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84451(Isoindoline, 18 | Isoindoline, 19)
Affinity DataKi:  0.600nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169842(1-(2,4-difluorophenethyl)-4-fluoro-4-(4-fluorophen...)
Affinity DataKi:  0.630nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169841(4-(4-Chloro-benzenesulfonyl)-1-[2-(2,4-difluoro-ph...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169844(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-[1...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169847(4-(4-Azetidin-1-yl-benzenesulfonyl)-1-[2-(2,4-difl...)
Affinity DataKi:  1nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  1nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84446(Isoindoline, 13)
Affinity DataKi:  1.20nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84443(Isoindoline, 10 | Isoindoline, 11)
Affinity DataKi:  1.20nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  1.33nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84453(Isoindoline, 20)
Affinity DataKi:  1.40nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169845(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(4-py...)
Affinity DataKi:  2nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169846(2-(4-Benzenesulfonyl-piperidin-1-yl)-1-(2,4-difluo...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169839(4-{1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-pipe...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84459(Isoindoline, 26)
Affinity DataKi:  3.60nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84449(Isoindoline, 16)
Affinity DataKi:  3.70nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84456(Isoindoline, 23)
Affinity DataKi:  4.10nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84448(Isoindoline, 15)
Affinity DataKi:  4.5nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84456(Isoindoline, 23)
Affinity DataKi:  5.30nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84446(Isoindoline, 13)
Affinity DataKi:  11.9nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84449(Isoindoline, 16)
Affinity DataKi:  12.4nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169840(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(2-fl...)
Affinity DataKi:  14nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84453(Isoindoline, 20)
Affinity DataKi:  17.5nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84459(Isoindoline, 26)
Affinity DataKi:  19nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84450(Isoindoline, 17)
Affinity DataKi:  19.1nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84451(Isoindoline, 18 | Isoindoline, 19)
Affinity DataKi:  20nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84447(Isoindoline, 14)
Affinity DataKi:  23nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84457(Isoindoline, 24)
Affinity DataKi:  24.3nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50108690(1-(2,4-difluorophenethyl)-4-(phenylsulfonyl)piperi...)
Affinity DataKi:  25nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84450(Isoindoline, 17)
Affinity DataKi:  26nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  35.4nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84443(Isoindoline, 10 | Isoindoline, 11)
Affinity DataKi:  35.9nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  43nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169848(1-[2-(2,4-Difluoro-phenyl)-ethyl]-4-fluoro-4-(3-fl...)
Affinity DataKi:  49nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169838(4-Benzenesulfonyl-1-[2-(2,4-difluoro-phenyl)-ethyl...)
Affinity DataKi:  49nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2c receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Aventis Pharmaceuticals

LigandPNGBDBM84440(Isoindoline, 7 | Isoindoline, 8 | Isoindoline, 9)
Affinity DataKi:  54.5nMAssay Description:All rat alpha-1 adrenoceptor binding was performed by Hugo M. vargas, Karen M. Brooks and Lynn Laws-Ricker.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Aventis Pharmaceuticals

LigandPNGBDBM84445(Isoindoline, 12)
Affinity DataKi:  55.9nMAssay Description:Dopamine D4.2 and D2S receptor binding was performed at NPS Allexlix Corp.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
University Of Uppsala

Curated by ChEMBL
LigandPNGBDBM50228614(CHEMBL51405)
Affinity DataKi:  56nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
University Of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004726(1-(1-Methyl-4-pyrrolidin-1-yl-but-2-ynyl)-pyrrolid...)
Affinity DataKi:  59nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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