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Found 341 with Last Name = 'vaudry' and Initial = 'h'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002726(CHEMBL2371933)
Affinity DataKi:  0.910nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002718(CHEMBL385281)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002725(CHEMBL374468)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002728(CHEMBL218825)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002723(CHEMBL265166)
Affinity DataKi:  2.40nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  2.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002717(CHEMBL216712)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002727(CHEMBL266651)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  4.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity against Human 5-HT7R expressed in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Binding affinity against Human 5-HT7R expressed in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210122(CHEMBL234881 | [2-(2',6'-dimethyl-biphenyl-3-yl)-e...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  6.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM50019568(Ala-Gly-c(Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210124(2-(2'-methyl-biphenyl-3-yl)-ethylamine | CHEMBL234...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210123(CHEMBL395870 | N,N-dimethyl-2-(2'-methylbiphenyl-3...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  8.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210126(CHEMBL232792 | [2-(2'-methoxy-biphenyl-3-yl)-ethyl...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  8.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50210125(CHEMBL232791 | [2-(2',6'-dimethoxy-biphenyl-3-yl)-...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002716(CHEMBL383996)
Affinity DataKi:  9.10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity against rat 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002719(CHEMBL412179)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD from human 5HT7 in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18nMAssay Description:Binding affinity against Human 5-HT7R expressed in sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18.5nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170159(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-p...)
Affinity DataKi:  18.5nMAssay Description:Binding affinity against rat 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  19nMAssay Description:Binding affinity against rat 5-HT7R expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002715(CHEMBL376223)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170158(1-(2-Methoxy-phenyl)-4-(1-o-tolyl-1H-pyrrol-3-ylme...)
Affinity DataKi:  21nMAssay Description:Binding affinity against rat 5-HT7R expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002720(CHEMBL219356)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  32.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  33.7nMAssay Description:Binding affinity to rat 5HT1AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170156(2-(3-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1...)
Affinity DataKi:  33.7nMAssay Description:Binding affinity against rat 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM85080(CH-275 | CH275 | L-Cys(1)-L-Lys-L-Phe-L-Phe-D-Trp-...)
Affinity DataKi:  45.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002724(CHEMBL428990)
Affinity DataKi:  74nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  83.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Université

Curated by ChEMBL
LigandPNGBDBM50170157(1-(2-Methoxy-phenyl)-4-[1-(2-trifluoromethyl-pheny...)
Affinity DataKi:  105nMAssay Description:Binding affinity against rat 5-HT7R expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002722(CHEMBL415851)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002713(CHEMBL425467)
Affinity DataKi:  155nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM82253(BIM 23052 | CAS_133073-82-2)
Affinity DataKi:  163nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Rouen

Curated by ChEMBL
LigandPNGBDBM50002698(CHEMBL437110)
Affinity DataKi:  263nMAssay Description:Displacement of [125I]human urotensin-2 from human GPR14 transfected in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM85080(CH-275 | CH275 | L-Cys(1)-L-Lys-L-Phe-L-Phe-D-Trp-...)
Affinity DataKi:  279nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(RAT)
Dynamique Des Systemes Neuroendocriniens

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  301nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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