TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 0.00200nMAssay Description:Competitive inhibition of DOT1L (2 to 416 residues) (unknown origin) using biotinylated nucleosomes as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase, H3 lysine-79 specific(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 0.0120nMAssay Description:Competitive inhibition of DOT1L (2 to 416 residues) (unknown origin) using biotinylated nucleosomes as substrate preincubated for 30 mins followed by...More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of 125-I echistatin from Vitronectin receptor (alpha v beta3)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of 125-I echistatin from Vitronectin receptor (alpha v beta3)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity to integrin alphavbeta3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity to GP2b3a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro activity in an vitronectin receptor (alpha v beta3) scintillation bead assay using 125-I labelled echistatin as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:Binding affinity to GP2b3a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity towards vitronectin receptor (alpha V-beta3) was determinedMore data for this Ligand-Target Pair