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Found 595 with Last Name = 'ventura' and Initial = 'm'
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205313(CHEMBL265859 | d[Leu4]AVP)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(CHEMBL375324 | d[Arg4]AVP)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205309(CHEMBL412972 | d[Leu4,Lys8]VP)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205296(CHEMBL385739 | d[Arg4,Dab8]VP)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205305(CHEMBL375324 | d[Arg4]AVP)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(CHEMBL221436 | d[Val4]AVP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205297(CHEMBL412973 | d[Leu4,Dab8]VP)
Affinity DataKi:  0.25nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205301(CHEMBL375188 | d[Leu4,Orn8]VP)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205304(CHEMBL435323 | dVDAVP)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205308((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205300(CHEMBL221436 | d[Val4]AVP)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004767(CHEMBL2312536)
Affinity DataKi:  0.309nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica

Curated by ChEMBL
LigandPNGBDBM50210579((2S,5S,8S,11R,13S,14S,17S,20S,23S)-23-amino-2-benz...)
Affinity DataKi:  0.310nMAssay Description:Inhibition of active BACE1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]-spiperone from D4 (unknown origin) receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50257034(CHEMBL4096543)
Affinity DataKi:  0.331nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  0.372nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205303(CHEMBL373968 | d[Leu4,Dap8]VP)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004768(CHEMBL2312538)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50401953(CHEMBL2207643)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205306(CHEMBL375323 | d[Orn4,Lys8]VP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205311(CHEMBL375096 | d[Orn4]AVP)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50608788(CHEMBL5285358)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50094505(2-((4-phenylpiperazin-1-yl)methyl)-1H-indole-5-car...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004766(CHEMBL2312226)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259021(CHEMBL4067083)
Affinity DataKi:  0.562nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004769(CHEMBL2312537)
Affinity DataKi:  0.589nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205292(CHEMBL385068 | d[Arg4,Orn8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205298(CHEMBL375325 | d[Arg4,Lys8]VP)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412783(CHEMBL493486)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259024(CHEMBL4071929)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50608785(CHEMBL5272162)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004770(CHEMBL2312227)
Affinity DataKi:  0.661nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259000(CHEMBL4082195)
Affinity DataKi:  0.692nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50608786(CHEMBL5278853)
Affinity DataKi:  0.760nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259023(CHEMBL4075507)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205307(CHEMBL412742 | d[Cha4,Dab8]VP)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259020(CHEMBL4091168)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205310(CHEMBL219272 | d[Orn4,Orn8]VP)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]AVP from rat vasopressin V1b receptor expressed in At-T20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50205291((S)-1-((4R,7S,10S,13S,16S)-7-(2-amino-2-oxoethyl)-...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50030196(CHEMBL3354065)
Affinity DataKi:  0.977nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50094503(2-((4-(4-fluorophenyl)piperazin-1-yl)methyl)-1H-in...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-spiperone from human D4 receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNischarin(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50259022(CHEMBL4070363)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor expressed in human HeLa cell membranes after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50004770(CHEMBL2312227)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha-1d adrenergic receptor expressed in CHO cell membranes after 30 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(RAT)
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]AVP from rat OT receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Instituto De Biologia Experimental E Tecnol£Gica

Curated by ChEMBL
LigandPNGBDBM50210579((2S,5S,8S,11R,13S,14S,17S,20S,23S)-23-amino-2-benz...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human recombinant BACE1 using Mca-SEVNLDAEFK-DNP substrate assessed as substrate hydrolysis after 2 hrs by HPLC-FLU analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026917(8-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-8-a...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]prazosin from recombinant human alpha-1d adrenergic receptor expressed in CHO cell membranes after 30 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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