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Found 282 with Last Name = 'vevert' and Initial = 'jp'
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50005878(4-Chloromethylsulfanyl-10,13-dimethyl-1,6,7,8,10,1...)
Affinity DataKi:  27nMAssay Description:Inhibition constant for human placental cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataKi:  27nMAssay Description:Inhibition constant for human placental cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50005876(4-Chloromethylsulfanyl-10,13-dimethyl-1,6,7,8,9,10...)
Affinity DataKi:  30nMAssay Description:Inhibition constant for human placental cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50005874(4-Fluoromethylsulfanyl-10,13-dimethyl-1,6,7,8,9,10...)
Affinity DataKi:  30nMAssay Description:Inhibition of cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50005875(4-Mercapto-10,13-dimethyl-1,6,7,8,10,12,13,14,15,1...)
Affinity DataKi:  72nMAssay Description:Inhibition constant for human placental cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Centre De Recherches Roussel-Uclaf

Curated by ChEMBL
LigandPNGBDBM50406730(CHEMBL2113619)
Affinity DataKi:  169nMAssay Description:Inhibition constant for human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285761(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285769(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285760(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285767(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.300nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285752(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.400nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285762(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285770(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285768(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50:  0.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285763(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.600nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285754(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.700nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093978(2-(4-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  0.810nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285762(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  0.900nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285764(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285752(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285763(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285757(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093996(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093987(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285753(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094000(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285755(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  1.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285758(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285754(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.10nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285758(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093985(2-(6-Carboxy-4H-benzo[1,3]dioxin-8-ylmethyl)-4-(6-...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093999(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093993(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  2.60nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285757(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.80nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285771(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  2.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093995(2-(2-Carboxymethoxy-cyclohexylmethyl)-4-(6-chloro-...)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093996(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093984(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  3.30nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094004(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.40nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093980(2-Adamantan-1-ylmethyl-4-(6-chloro-benzo[1,3]dioxo...)
Affinity DataIC50:  3.40nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093993(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.60nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50285756(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.80nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50285766(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285770(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  3.90nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093988(2-(2-Carboxymethoxy-4-methoxy-benzyl)-4-(6-chloro-...)
Affinity DataIC50:  4nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093986(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  4.60nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285766(5-alpha-hydroxyacid imidazolyl biphenyl sulfonyl u...)
Affinity DataIC50:  4.70nMAssay Description:In vitro binding affinity at Angiotensin II Type 2 receptor in rabbit uterus membrane by [125I]-AII displacement.More data for this Ligand-Target Pair
In DepthDetails Article
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