Affinity DataKi: 0.790nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 2.22nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 2.25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 4.26nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 5.04nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 5.63nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 9.02nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 26.2nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 42.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 53.1nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 76.8nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
The Walter And Eliza Hall Institute Of Medical Research
Curated by ChEMBL
The Walter And Eliza Hall Institute Of Medical Research
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 128nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 150nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetCytochrome P450 3A4(Homo sapiens (Human))
The Walter And Eliza Hall Institute Of Medical Research
Curated by ChEMBL
The Walter And Eliza Hall Institute Of Medical Research
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2B receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 243nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 245nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2B receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Binding affinity to adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A3 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Antagonist activity rat recombinant GluN1/GluN2C receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response by...More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University (Parkville Campus)
Curated by ChEMBL
Monash University (Parkville Campus)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Displacement of [125I]ABA from human recombinant adenosine A1 receptor by rapid filtration techniqueMore data for this Ligand-Target Pair