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Found 29 with Last Name = 'visan' and Initial = 'v'
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)
Affinity DataIC50:  10nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50:  20nMAssay Description:Inhibition of IK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)
Affinity DataIC50:  70nMAssay Description:Inhibition of IK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279024((1,3-dimethyl-1H-pyrazol-5-yl)(5-(furan-2-carbonyl...)
Affinity DataIC50:  710nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278971(2-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278972(CHEMBL500166 | methyl 2-(5-(furan-2-carbonyl)-5,6-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278973((5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6-y...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278994(CHEMBL498728 | phenanthridine-5,6(6H)-diylbis(fura...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278938(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279105(5-(3-chlorobenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279066(5-(3-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278939((6-(cyclobutanecarbonyl)phenanthridin-5(6H)-yl)(fu...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279107(1-((2-chlorophenyl)diphenylmethyl)-1H-pyrazole | C...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278936(1-(6-(1H-indol-3-yl)phenanthridin-5(6H)-yl)ethanon...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279063(5-tosyl-5H-dibenzo[b,d]azepin-7(6H)-one | CHEMBL49...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279065(5-(4-chlorophenylsulfonyl)-5H-dibenzo[b,d]azepin-7...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50278937(1-(5-(furan-2-carbonyl)-5,6-dihydrophenanthridin-6...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279064(5-(4-nitrophenylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50279104(5-(4-methylbenzoyl)-5H-dibenzo[b,d]azepin-7(6H)-on...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed