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Found 930 with Last Name = 'visser' and Initial = 's'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50088475(1-(2-Methoxy-phenyl)-3-(2-pyridin-3-yl-quinazolin-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097451(4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067116(4-Methoxy-N-(3-pyridin-2-yl-isoquinolin-1-yl)-benz...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097441(4-Methoxy-N-(2-phenyl-quinazolin-4-yl)-benzamide |...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097436(4-Methyl-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097440(CHEMBL165783 | N-(3-Phenyl-[1,2,4]thiadiazol-5-yl)...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097432((Cis)-4-Methoxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097442(4-Chloro-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426((Cis)-4-Hydroxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097426((Cis)-4-Hydroxy-cyclohexanecarboxylic acid (3-phen...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide | 4-...)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097446(4-Methoxy-N-(3-phenyl-isoquinolin-1-yl)-benzamide ...)
Affinity DataKi:  79nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097452(CHEMBL354004 | [4-(3-Phenyl-[1,2,4]thiadiazol-5-yl...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097451(4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067081(9-Fluoro-2-furan-2-yl-5,6-dihydro-[1,2,4]triazolo[...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097436(4-Methyl-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50059376(9-Methyl-2-phenyl-5,9-dihydro-[1,2,4]triazolo[5,1-...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067096(CHEMBL71053 | N-(3-(pyridin-2-yl)isoquinolin-1-yl)...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097448(4-Chloro-N-(4-pyridin-2-yl-thiazol-2-yl)-benzamide...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097421(4-Methoxy-N-(6-phenyl-pyrimidin-4-yl)-benzamide | ...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067107(CHEMBL424259 | N-(2-Pyridin-2-yl-quinazolin-4-yl)-...)
Affinity DataKi:  230nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097434(CHEMBL435866 | N-(2-Phenyl-quinazolin-4-yl)-benzam...)
Affinity DataKi:  240nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097440(CHEMBL165783 | N-(3-Phenyl-[1,2,4]thiadiazol-5-yl)...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097442(4-Chloro-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benza...)
Affinity DataKi:  520nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097451(4-Hydroxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]-CGS-21,680 or [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097455(4-Methoxy-3-methyl-N-(3-phenyl-[1,2,4]thiadiazol-5...)
Affinity DataKi:  580nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097431(4-Methoxy-N-(4-phenyl-thiazol-2-yl)-benzamide | 4-...)
Affinity DataKi:  670nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097421(4-Methoxy-N-(6-phenyl-pyrimidin-4-yl)-benzamide | ...)
Affinity DataKi:  800nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097425(1-Phenyl-3-(4-pyridin-2-yl-thiazol-2-yl)-urea | CH...)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]-CGS-21,680 or [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097445(CHEMBL162808 | Cyclopentanecarboxylic acid (4-pyri...)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097425(1-Phenyl-3-(4-pyridin-2-yl-thiazol-2-yl)-urea | CH...)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097422(1-Phenyl-3-(3-phenyl-[1,2,4]thiadiazol-5-yl)-urea ...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097449(4-Iodo-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benzami...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097452(CHEMBL354004 | [4-(3-Phenyl-[1,2,4]thiadiazol-5-yl...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097439(CHEMBL163248 | N-(3-Phenyl-isoquinolin-1-yl)-benza...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097439(CHEMBL163248 | N-(3-Phenyl-isoquinolin-1-yl)-benza...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097445(CHEMBL162808 | Cyclopentanecarboxylic acid (4-pyri...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]-CGS-21,680 or [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097444(3-Chloro-N-(4-pyridin-2-yl-thiazol-2-yl)-benzamide...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]-CGS-21,680 or [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097428(CHEMBL164782 | Cyclohexanecarboxylic acid (3-pheny...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097429(4-Nitro-N-(4-pyridin-2-yl-thiazol-2-yl)-benzamide ...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097443(4-Methyl-N-(4-pyridin-2-yl-thiazol-2-yl)-benzamide...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50097450(3,4-Dichloro-N-(4-pyridin-2-yl-thiazol-2-yl)-benza...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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