TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 398nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 501nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 794nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of GST-tagged human BRD3 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human BRD3 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of GST-tagged human BRD3 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human BRD3 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of TEV cleavage site-fused-GST tagged BRD4(BD1) (unknown origin) using SGRGK(Ac)CGK(Ac)-GLGK(Ac)GGAK(Ac)RHRKVG-peptide after 3 hrs by HTRF...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.64E+4nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 3.17E+4nMAssay Description:Inhibition of GST-tagged human BRD3 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of GST-tagged human BRD4 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of GST-tagged human BRD2 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of GST-tagged human BRD3 bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain testis-specific protein(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged human BRDT bromodomain1 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetATPase family AAA domain-containing protein 2(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GST-tagged human ATAD2 using H4KAc 5/8/12/16 peptide as substrate incubated overnight by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataKd: 540nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataKd: 410nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataKd: 320nMAssay Description:Binding affinity to TEV cleavage site-fused-His-tagged BRD4(BD1) (unknown origin) by isothermal-titration calorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Aix-Marseille University
Curated by ChEMBL
Aix-Marseille University
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to his-tagged human BRD4 bromodomain1 by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair