TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: <0.5nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: <0.5nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.610nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of recombinant JAK2 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory constant against Serotonin transporterMore data for this Ligand-Target Pair
Affinity DataIC50: 34.1nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 41.5nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 175nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 178nMAssay Description:Inhibition of recombinant ABL1 T315I mutant (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant ABL1 T315I mutant (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Beckman Research Institute
Curated by ChEMBL
Beckman Research Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant GST-tagged c-Src (unknown origin) expressed in insect cells using pEY as substrate preincubated with enzyme followed by [33...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 224nMAssay Description:Inhibition of recombinant JAK2 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant c-Src (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 468nMAssay Description:Inhibition of recombinant ABL1 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 551nMAssay Description:Inhibition of recombinant JAK2 (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 589nMAssay Description:Inhibition of recombinant Aurora A (unknown origin) after 120 mins in presence of [33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair