TargetMultidrug and toxin extrusion protein 1(Mus musculus)
Riken Center For Life Science Technologies
Curated by ChEMBL
Riken Center For Life Science Technologies
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Inhibition of mouse Mate1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analy...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 1(Mus musculus)
Riken Center For Life Science Technologies
Curated by ChEMBL
Riken Center For Life Science Technologies
Curated by ChEMBL
Affinity DataKi: 3.60E+3nMAssay Description:Inhibition of mouse Oct1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analys...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of specific binding of [3H]BK at 0.06 nM to bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:In vitro inhibitory activity towards bradykinin receptor B2 using [3H]BK (0.06 nM) as a radioligand in guinea pig ileum membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%.More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Mochida Pharmaceutical
US Patent
Mochida Pharmaceutical
US Patent
Affinity DataIC50: <0.100nMAssay Description:Measurement was carried out using TrkA LanthaScreen (registered trademark) Eu Kinase Binding Assay (ThermoFisher SCIENTIFIC). To a 384 well plate (Co...More data for this Ligand-Target Pair
Ligand Info