Affinity DataKi: 111nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 751nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.45E+3nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 3.58E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 6.78E+3nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 1.03E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+4nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 1.78E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 1.96E+4nMAssay Description:Invitro inhibition was measured against Bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 2.51E+4nMAssay Description:Invitro inhibition was measured against Human bovine pancreatic trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >3.37E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: >3.37E+4nMAssay Description:Invitro inhibition was measured against Human Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 6.24E+4nMAssay Description:Invitro inhibition was measured against Human Thrombin.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of PRMT5 in human HCT116-MTAP null cells assessed as reduction in symmetric dimethylation of arginine using SAM as substrate incubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of PRMT5 in human HCT116-MTAP null cells assessed as reduction in symmetric dimethylation of arginine using SAM as substrate incubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against human fibroblast collagenase (MMP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against human fibroblast collagenase (MMP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged MAT2A expressed in Escherichia coli using methionine and ATP as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged MAT2A expressed in Escherichia coli using methionine and ATP as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of PRMT5 in human HCT116-MTAP null cells assessed as reduction in symmetric dimethylation of arginine using SAM as substrate incubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged MAT2A expressed in Escherichia coli using methionine and ATP as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged MAT2A expressed in Escherichia coli using methionine and ATP as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of full length recombinant human N-terminal His6-tagged MAT2A expressed in Escherichia coli using methionine and ATP as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 24nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of PRMT5 in human HCT116-MTAP null cells assessed as reduction in symmetric dimethylation of arginine using SAM as substrate incubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against human fibroblast collagenase (MMP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against human fibroblast collagenase (MMP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMpH: 7.5 T: 2°CAssay Description:Assays were performed in 96-well microtiter plates in reaction buffer containing biotinylated substrate, ATP/[gamma-33P]ATP, and purified kinase in t...More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Compound was tested for its inhibitory activity against 92 kD gelatinase (MMP-9)More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against human fibroblast collagenase (MMP-1)More data for this Ligand-Target Pair