TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 47.6nMAssay Description:Inhibitory activity against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:Inhibitory activity of the compound against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 97.8nMAssay Description:Inhibitory activity of the compound against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 98nMAssay Description:Inhibitory activity against CCR5 receptor in CHO cell membranes was determined using radio-ligand [125I]-RANTES binding assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 5.10E+3nMAssay Description:Inhibitory activity of the compound against human CCR5 chemokine receptor (CCR5) expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M2(RAT)
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 3.00E+4nMAssay Description:Inhibitory activity of the compound against human CCR5 chemokine receptor (CCR5) expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Mus musculus)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to muscarinic receptor in miceMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]-DTG from sigma opioid receptor of homogenized guinea pig whole brainMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions
Curated by ChEMBL
Johns Hopkins Medical Institutions
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair