Affinity DataKi: 1.00E+8nMAssay Description:Inhibition of 5HT6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+8nMAssay Description:Inhibition of 5HT3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+8nMAssay Description:Inhibition of histamine H2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+8nMAssay Description:Inhibition of 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human P2X2/3 receptor expressed in 1321n1c cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of P2X2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat P2X3 receptor expressed in CHO cells by FLIPRMore data for this Ligand-Target Pair